1. GPCR/G Protein
  2. Adenosine Receptor

GR79236 

Cat. No.: HY-18978
Handling Instructions

GR79236 is a highly potent and selective adenosine A1 receptor agonist (Ki = 3.1 nM) that has analgesic and anti-inflammatory actions in humans and animals.

For research use only. We do not sell to patients.
GR79236 Chemical Structure

GR79236 Chemical Structure

CAS No. : 124555-18-6

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Free Sample (0.5-1 mg)   Apply now  
10 mM * 1 mL in Water $99 In-stock
5 mg $90 In-stock
10 mg $120 In-stock
50 mg $480 In-stock
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  • Biological Activity

  • Technical Information

  • References

Description

GR79236 is a highly potent and selective adenosine A1 receptor agonist (Ki = 3.1 nM) that has analgesic and anti-inflammatory actions in humans and animals. IC50 value: 3.1 nM(Ki) Target: adenosine A1 receptor in vitro: GR79236 is a highly potent and selective A1-receptor agonist that is originally developed for the treatment of Type 2 diabetes mellitus, as a cardioprotective agent and also for peripheral arterial occlusive diseases. in vivo: GR79236 has also been shown to have antinociceptive and anti-inflammatory properties in animal models. GR79236 inhibits the release of CGRP evoked by superior sagittal sinus (SSS) stimulation in the cat and inhibits trigeminal nucleus firing in the cat and rat. GR79236X has acute, short-term analgesic efficacy.

References
Molecular Weight

351.36

Formula

C₁₅H₂₁N₅O₅

CAS No.

124555-18-6

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

Solvent & Solubility

H2O: ≥ 100 mg/mL

* "<1 mg/mL" means slightly soluble or insoluble. "≥" means soluble, but saturation unknown.

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GR79236
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HY-18978
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