1. GPCR/G Protein
  2. P2Y Receptor
  3. Prasugrel (Maleic acid)

Prasugrel (Maleic acid) (Synonyms: PCR 4099 (Maleic acid))

Cat. No.: HY-15284B
Handling Instructions

Prasugrel (PCR 4099) Maleic acid is a thienopyridine and prodrug, inhibits platelet function. Prasugrel Maleic acid is an orally active and potent P2Y12 receptor antagonist, and inhibits ADP-induced platelet aggregation.

For research use only. We do not sell to patients.

Prasugrel (Maleic acid) Chemical Structure

Prasugrel (Maleic acid) Chemical Structure

CAS No. : 389574-20-3

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Description

Prasugrel (PCR 4099) Maleic acid is a thienopyridine and prodrug, inhibits platelet function. Prasugrel Maleic acid is an orally active and potent P2Y12 receptor antagonist, and inhibits ADP-induced platelet aggregation[1].

IC50 & Target

P2Y12 receptor[1]

In Vitro

In rat platelets, Prasugrel (PCR 4099) Maleic acid active metabolite inhibits in vitro platelet aggregation induced by adenosine ADP (10μM) with an IC50 value of 1.8 μM[2].
Prasugrel (PCR 4099) Maleic acid acts faster and is significantly more potent than Clopidogrel in vivo. Prasugrel hydrochloride is an inactive prodrug that requires metabolic processing in vivo to generate the active antiplatelet metabolite. Prasugrel (PCR 4099) Maleic acid is rapidly absorbed from the gut. After oral administration of standard-loading doses of 60 mg, maximum plasma levels of the active metabolite are achieved within 1 h, effective, maximum inhibition of platelet aggregation at 1-2 h[1].

Clinical Trial
Molecular Weight

489.51

Formula

C₂₄H₂₄FNO₇S

CAS No.

389574-20-3

SMILES

O=C(O)/C=C\C(O)=O.FC1=CC=CC=C1C(C(C2CC2)=O)N3CCC4=C(C3)C=C(S4)OC(C)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

Prasugrel (Maleic acid)PCR 4099 (Maleic acid)P2Y ReceptoractivemetaboliteantiplateletADPplateletaggregationInhibitorinhibitorinhibit

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Prasugrel (Maleic acid)
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