BChE-IN-36
hBChE-IN-4 (compound 40) is a potent hCA activator and BChE inhibitor with KA values of 266, 76.9, 918, 893, 98.0 nM for hCA I, hCA II, hCA IV, hCA VB, hCA VII, IC50 values of 72.1, 4.2 nM for eeAChE, eqBChE, respectively. hBChE-IN-4 shows no cytotoxicity. hBChE-IN-4 shows potent procognitive effects. hBChE-IN-4 has the potential for the research of neurodegenerative diseases and other neuropsychiatric disorders.
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- Formule: C26H35N5O2
- Masse moléculaire:449.59
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
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EeAChE 72.1 nM (IC50) |
eqBCHE 4.2 nM (IC50) |
hCA I 266 nM (KA) |
hCA II 76.9 nM (KA) |
hCA VB 893 nM (KA) |
hCA IV 918 nM (KA) |
hCA VII 98.0 nM (KA) |
Chemical Information
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Masse moléculaire 449.59
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Formule C26H35N5O2
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SMILES
O=C([C@@H](NCCCCCCNC1=C2CCCCC2=NC3=CC=CC=C31)CC4=CNC=N4)OC
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
BChE-IN-36 Related Classifications
HY-169163 Related Classifications
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