A3AR antagonist-7
A3AR antagonist-7 is a conjugable human A3 adenosine receptor (A3AR) antagonist with a Ki value of 31.8 nM. A3AR antagonist-7 is applicable to the research of melanoma, breast cancer and colorectal cancer.
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- CAS No.: 2672534-18-6
- Formule: C56H71N15O12S2
- Masse moléculaire:1210.39
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
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Activité biologique
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Adenosine A3 receptor 31.8 nM (Ki) |
A3AR antagonist-7 (Compound 23) binds to hA3AR expressed in CHO cells with a Ki of 31.8 nM, shows lower affinity for hA2AAR expressed in HEK293 cells (Ki = 90 nM), and has undetermined binding to hA1AR expressed in CHO cells, with a hA2AAR/hA3AR selectivity ratio of 2.83[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2672534-18-6
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Masse moléculaire 1210.39
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Formule C56H71N15O12S2
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SMILES
O=C(C1=C(C2=C(C=CC(N)=C3S(=O)(O)=O)C3=[O+]C4=C2C=CC(N)=C4S(=O)(O)=O)C=CC(C(NCCCCCCN5N=NC(CCCC(NC6=NC7=NN(C)C=C7C8=NC(C9=CC=CO9)=NN68)=O)=C5)=O)=C1)[O-].CCN(CC)CC.CCN(CC)CC
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
A3AR antagonist-7 Related Classifications
HY-182432 Related Classifications
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