YM218 free base
YM218 free base is an orally active non-peptide vasopressin (AVP) receptor antagonist. YM218 free base has a high affinity for rat liver V1A receptors with a Ki value of 0.50 nM; it has a lower affinity for rat pituitary V1B, kidney V2, and uterine oxytocin receptors with Ki values of 1510 nM, 72.2 nM, and 150 nM, respectively. YM218 free base can be used in the study of diabetes and kidney disease.
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- CAS No.: 387816-81-1
- Formule: C35H38F2N4O4
- Masse moléculaire:616.70
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
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Activité biologique
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Rat liver V1a Receptor 0.5 nM (Ki) |
Rat pituitary V1b receptor 1510 nM (Ki) |
Rat kidney V2 receptor 72.2 nM (Ki) |
Chemical Information
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CAS No. 387816-81-1
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Masse moléculaire 616.70
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Formule C35H38F2N4O4
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SMILES
O=C(NC1=CC=C(C=C1)C(N2CCC(F)(/C(C3=CC=CC=C32)=C\C(N4CCC(CC4)N5CCCCC5)=O)F)=O)C6=C(OC=C6)C
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
YM218 free base Related Classifications
HY-118918 Related Classifications
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