Copy Link Print Information

G15

41 Cited Publications
Customer Review

Based on 41 publication(s) in Google Scholar

G15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM.

For research use only. We do not sell to patients.

  • Purity: 99.0%
  • CAS No.: 1161002-05-6
  • Formula: C19H16BrNO2
  • Molecular Weight:370.24
  • Storage:

    -20°C, protect from light

    * In solvent : -80°C, 2 years; -20°C, 1 year (protect from light)

  • G15 Chemical Structure
    G15 Chemical Structure
  • Experimental Validation Results for G15
  • Experimental Validation Results for G15
  • Experimental Validation Results for G15
  • Experimental Validation Results for G15
  • Experimental Validation Results for G15
CAS No.: 1161002-05-6
Size
Price
Stock
Quantity
Amount: USD 0.00
Please select quantity
or
or

* Please select Quantity before adding items.

To place orders, for customer services and technical support, please contact: MedChemExpress USA

Tel: 609-228-6898 E-mail: [email protected] [email protected]

Data Download
Other Forms of G15:

To place orders, for customer services and technical support, please contact:

609-228-6898
[email protected] [email protected]
Find Your Local Distributor Your local distributor: Hycultec GmbHHycultec
  • Biological Activity
  • Chemical Information
  • Solvent & Solubility
  • Purity & Documentation
  • References
  • Help & FAQs
You May Still Need
Top Publications Citing

Use of MCE Products

Publications Citing Use of MedChemExpress (MCE) G15

More
Customer Validation & Images
WBOthersRT-PCRCell Imaging/Staining
  • RT-PCR
  • Others
  • WB
  • WB
  • Cell Imaging/Staining

All Estrogen Receptor/ERR Isoforms

More
Keywords
100 mg

Get Quote In-stock

Please select quantity
Amount: USD 0.00
Sign in to MedChemExpress Sign In
Register
Sign in to MedChemExpress
Register New Account

At least 6 characters

Personalize your experience, you are currently not signed in. For a better experience, please create an online profile, you can:

Obtain points redemption prizes
Check out faster
Add multiple shipping locations
View orders
Assay Types
  • G15 Chemical Structure
    G15 Chemical Structure
    1/16
  • 1/16

    G15 purchased from MedChemExpress. Usage Cited in: Poult Sci. 2025 Dec 5;105(1):106210. [Abstract]

    Customer Validation
     Effects of selective receptor agonists (PPT, DPN and G-1) treatment (3 h) on PGR expression, and antagonist (ICI and G15) treatment (3 h) on E2-upregulated PGR expression, in cultured pituitary cells from female chicks.

  • 1/16

    G15 purchased from MedChemExpress. Usage Cited in: Pharm Biol. 2023 Dec;61(1):499-513. [Abstract]

    Customer Validation
     TMYX enhanced the dilation function of coronary microvessels in vitro, but this effect was inhibited by G-15.

  • 1/16

    G15 purchased from MedChemExpress. Usage Cited in: Cell Death Dis. 2022 Apr 19;13(4):372. [Abstract]

    Customer Validation
     J774A.1 cells were pre-treated with DHEA (50 μM) in the presence or absence of the GPER inhibitor G15 (1 μM) for 1 h, then stimulated with LPS for 4 h. The TLR4, p-ERK/ERK, LC3, p62, p-mTOR, and p-AMPK protein expression levels were measured by western blotting and quantified by Image J software.

  • 1/16

    G15 purchased from MedChemExpress. Usage Cited in: Cell Death Dis. 2022 Apr 19;13(4):372. [Abstract]

    Customer Validation
     J774A.1 cells were pre-treated with G1 (1 μM) for 1 h, then stimulated with LPS for 4 h, and the indicated protein expression levels were measured by western blotting and quantified by Image J software.

  • 1/16

    G15 purchased from MedChemExpress. Usage Cited in: Cell Death Dis. 2022 Apr 19;13(4):372. [Abstract]

    Customer Validation
     J774A.1 cells were pre-treated with DHEA (50 μM) in the presence or absence of the GPER inhibitor G15 (1 μM) for 1 h, then stimulated with LPS for 4 h, PI-positive dead cells in 5 randomly selected fluorescence microscope images were counted by Image J software, scale bar = 200 μm.

  • G15