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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
20 Results for "
Apalutamide
" in MedChemExpress (MCE) Product Catalog:
Products (20)
20 Results for "Apalutamide" in MCE Product Catalog:
15
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Apalutamide (ARN-509) is a potent and competitive androgen receptor (AR) antagonist, binding AR with an IC50 of 16 nM .
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1 Cited Publications
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N-Desmethyl-Apalutamide, the major active metabolite of Apalutamide (HY-16060), is a selective competitive inhibitor of androgen receptor. N-Desmethyl-Apalutamide is catalyzed by CYP3A4 and CYP2C8 enzymes. The plasma protein binding rate of N-Desmethyl-Apalutamide reaches 95%, with albumin as the primary binding protein. N-Desmethyl-Apalutamide is suitable for prostate cancer-related research .
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1
1 Cited Publications
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Apalutamide-COOH is a metabolite of Apalutamide. Apalutamide is a potent and competitive androgen receptor (AR) antagonist, binding AR with an IC50 of 16 nM .
Cat. No.: HY-P4070
CAS No.: 1188379-43-2
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Cat. No.: HY-16060S
CAS No.: 1638885-65-0
Synonyms: ARN-509-d4
Cat. No.: HY-W754151
Cat. No.: HY-16060S1
CAS No.: 1638885-61-6
Synonyms: ARN-509-d3
Cat. No.: HY-16060R
CAS No.: 956104-40-8
Synonyms: ARN-509 (Standard)
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Apalutamide (Standard) is the analytical standard of Apalutamide. This product is intended for research and analytical applications. Apalutamide (ARN-509) is a potent and competitive androgen receptor (AR) antagonist, binding AR with an IC50 of 16 nM .
Cat. No.: HY-16060S3
Synonyms: ARN-509-d7
Cat. No.: HY-16060S2
Synonyms: ARN-509-13C,d3
Cat. No.: HY-135331S
Cat. No.: HY-P11293
CAS No.: 1309855-53-5
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Cat. No.: HY-P4757
CAS No.: 108081-77-2
Cat. No.: HY-P1321
CAS No.: 158859-98-4
Synonyms: 1229U91; GW1229
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Cat. No.: HY-136596R
CAS No.: 1332391-04-4
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Nortriptyline (Standard) is the analytical standard of Nortriptyline. This product is intended for research and analytical applications. Nortriptyline (Desmethylamitriptyline), the main active metabolite of Amitriptyline, is a tricyclic antidepressant. Nortriptyline is a potent autophagy inhibitor and has anticancer effects .
N
Cat. No.: HY-P1321A
Synonyms: 1229U91 TFA; GW1229 TFA
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Cat. No.: HY-P11480
CAS No.: 3105660-96-3
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Cat. No.: HY-P12133
CAS No.: 3080063-21-1
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Tapimtrutide is a gastric inhibitory polypeptide (GIP) and glucagon-like peptide 1 (GLP-1) receptor agonist. Tapimtrutide can be used for the research of diabetes .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
