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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
46 Results for "
Cys491
" in MedChemExpress (MCE) Product Catalog:
Products (46)
46 Results for "Cys491" in MCE Product Catalog:
3
3 Cited Publications
Cat. No.: HY-P0171
CAS No.: 664334-36-5
Synonyms: BKT140 (4-fluorobenzoyl); BL-8040; TF14016
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2
2 Cited Publications
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Cardiovascular Disease Inflammation/Immunology Endocrinology
1
Lirafugratinib (RLY-4008) is an orally active, irreversible and highly selective FGFR2 inhibitor with an IC50 of 3 nM. Lirafugratinib covalently binds to Cys491. Lirafugratinib targets FGFR2 primary alterations and resistance mutations and induces tumor regression while sparing other FGFRs .
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1 Cited Publications
Synonyms: RLY-4008 hydrochloride
Lirafugratinib (RLY-4008) hydrochloride is an orally active, irreversible and highly selective FGFR2 inhibitor with an IC50 of 3 nM. Lirafugratinib hydrochloride covalently binds to Cys491. Lirafugratinib hydrochloride targets FGFR2 primary alterations and resistance mutations and induces tumor regression while sparing other FGFRs .
1
1 Cited Publications
Cat. No.: HY-P1604
CAS No.: 60748-45-0
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1 Cited Publications
Cat. No.: HY-P1604A
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Cat. No.: HY-12554
CAS No.: 14636-12-5
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Cardiovascular Disease Inflammation/Immunology Endocrinology
Terlipressin is a vasopressin analogue with potent vasoactive properties. Terlipressin is a highly selective vasopressin V1 receptor agonist that reduces the splanchnic blood flow and portal pressure and controls acute variceal bleeding. Terlipressin exerts anti-inflammatory and anti-oxidative effects. Terlipressin has the potential for hepatorenal syndrome and norepinephrine-resistant septic shock research .
Cat. No.: HY-P3732
CAS No.: 332179-76-7
Cat. No.: HY-P3499
CAS No.: 1092457-65-2
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Cat. No.: HY-P3099
CAS No.: 154525-25-4
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Cat. No.: HY-P1443
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Cat. No.: HY-P5174
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Cat. No.: HY-P5681
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Cat. No.: HY-P3912A
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Cat. No.: HY-P1457
CAS No.: 154765-05-6
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Cat. No.: HY-P3099A
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Cat. No.: HY-P5077A
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
