2 Results for "

HDAC-IN-30

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "HDAC-IN-30" in MCE Product Catalog:

Cat. No.: HY-144292
CAS No.: 2756809-34-2
Target:  

HDAC

Research Areas:  

Cancer

HDAC-IN-30 is a novel multi-target HDAC inhibitor, including HDAC1 (IC50=13.4 nM),HDAC2 (IC50=28.0 nM), HDAC3 (IC50=9.18 nM), HDAC6 (IC50=42.7 nM), HDAC8 (IC50=131 nM). HDAC-IN-30 exhibits potent antitumor efficacy .
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Cat. No.: HY-162349
CAS No.: 3030144-11-4
Target:  

HDAC PARP

Research Areas:  

Cancer

PARP7/HDACs-IN-1 (compound 9l) is a dual-target inhibitor targeting PARP7/HDAC with anti-tumor activity. PARP7/HDACs-IN-1 inhibits different subtypes of PARPs and HDACs with IC50s of 83.3 nM (PARP1), 3.1 nM (PARP7), 35 nM (HDAC1), 30.3 nM (HDAC2), 35.4 nM (HDAC3), and 6.4 nM respectively. (HDAC6) . br/ .
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