10 Results for "

hallucinogen

" in MedChemExpress (MCE) Product Catalog:
Products (10)

10 Results for "hallucinogen" in MCE Product Catalog:

Cat. No.: HY-100845
CAS No.: 83729-01-5
Synonyms: Divinorin A
Salvinorin A is a potent, unique and short-acting high efficacy kappa-opioid receptor (KOPr) agonist with Ki value of 4.3 nm. Salvinorin A is a non-nitrogenous neoclerodane isolated from Salvia divinorum.
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Cat. No.: HY-138218
CAS No.: 3270-02-8
Synonyms: 1-Acetyl-LSD
Research Areas:  

Neurological Disease

ALD-52 (1-Acetyl-LSD) is a prodrug for LSD. ALD-52 shows an affinity to 5-HT1A, 5-HT2A and 5-HT2C with a sub>D values of 1054, 174 and 10.2 nM, respectively. ALD-52 is converted to LSD and induces a head-twitch response (HTR) in vivo. ALD-52 can be used for hallucinogen research .
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Cat. No.: HY-130394
CAS No.: 178557-21-6
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

2C-B-FLY hydrochloride is the dihydrodifuran analog of the Schedule I hallucinogen 4-bromo-2,5-dimethoxyphenethylamine (2C-B).
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Cat. No.: HY-W742532
CAS No.: 65527-62-0
Synonyms: N-Ethyl-nor-LSD
Research Areas:  

Neurological Disease

ETH-LAD (N-Ethyl-nor-LSD) is an activator for 5-HT2A receptor with Ki of 5.1 nM. ETH-LAD exhibits affinity for dopamine receptor D1 and dopamine receptor D2 with Ki of 22.1 nM and 4.4 nM. ETH-LAD acts as psychoactive substance in rat model .
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Cat. No.: HY-Z8487
CAS No.: 1823362-29-3
Target:  

Drug Derivative

Research Areas:  

Neurological Disease

2-(2-Chlorophenyl)-2-hydroxycyclohexanone is structurally similar to known hallucinogens that is an impurity in Esketamine preparations .
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Cat. No.: HY-137920
CAS No.: 689295-71-4
Target:  

Opioid Receptor

Research Areas:  

Cardiovascular Disease

Salvinorin A (Divinorin A) propionate is a potent, unique and short-acting high efficacy kappa-opioid receptor (KOPr) agonist with Ki value of 4.3 nm. Salvinorin A propionate is a non-nitrogenous neoclerodane isolated from Salvia divinorum .
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Cat. No.: HY-170053
CAS No.: 763035-03-6
Synonyms: 4-OH-MPT; Meprocin
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

4-Hydroxy MPT (4-OH-MPT), a serotonergic hallucinogen, is a 5-HT2A and 5-HT2B receptors agonist with EC50 values of 3.82 nM and 3.4 nM, respectively .
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Cat. No.: HY-180584
CAS No.: 1555334-81-0
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

5-HT2A agonist 9 (Compound I-53) is a 5-HT2A agonist with an EC₅₀ of 34 nM. 5-HT2A agonist 9 can be used for the study of mental disorders and central system disorders .
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Cat. No.: HY-L121
427 compounds

5-HT receptors, also called Serotonin receptors, are a group of G protein-coupled receptors (GPCRs) and ligand-gated ion channels (LGICs) found in the central and peripheral nervous systems. These receptors are now classified into seven families, 5-HT1–7, comprising a total of 14 structurally and pharmacologically distinct mammalian 5-HT receptor subtypes. The 5-HT receptors influence various biological and neurological processes such as aggression, anxiety, appetite, cognition, learning, memory, mood, nausea, sleep, andthermoregulation. The serotonin receptors are the target of a variety of pharmaceutical drugs, including many antidepressants, antipsychotics, anorectics, antiemetics, gastroprokinetic agents, antimigraine agents, hallucinogens, and entactogens.

MCE 5-HT Receptor Compound Library consists of 427 5-HT receptor inhibitors and activators, which can be used for neuropsychiatric disorders drugs discovery.

Cat. No.: HY-N20747
CAS No.: 28363-70-4
Synonyms: 4-Hydroxy-N-methyltryptamine; 4-HO-NMT
Norpsilocin (4-hydroxy-N-methyltrypt amine; 4-HO-NMT) is a natural tryptamine alkaloid isolated from the hallucinogenic mushroom Psilocybe cubensis. Norpsilocin activates human 5-HT2 receptors (5-HT2A: EC50 = 8.4 nM; 5-HT2B = 12.8 nM; 5-HT2C = 39.6 nM) and displays binding affinity toward 5-HT1 receptors (5-HT1B: Ki = 212 nM; 5-HT1D = 48.9 nM; 5-HT1E = 81.7 nM). Norpsilocin induces β-arrestin recruitment at the 5-HT1B receptor. Norpsilocin fails to produce psychedelic-like effects in mice, whereas high doses can induce hypothermia in vivo. Norpsilocin acts as an important research tool for exploring the structure–activity relationship of tryptamine hallucinogens and the pharmacology of serotonin receptors .
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