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MRS8454

MRS8454 is a positive allosteric modulator (PAM) of the A3 adenosine receptor (A3AR). MRS8454 can significantly enhance the maximum effect of the standard agonist Cl-IB-MECA by approximately 286%-300%, and significantly reduce its EC50 value. MRS8454 effectively enhances the ability of A3AR agonists to inhibit the cAMP accumulation induced by Forskolin (HY-15371). MRS8454 can be used for the development of molecular probes.

For research use only. We do not sell to patients.

  • Formula: C46H59N5
  • Molecular Weight:681.99
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

  • MRS8454 Chemical Structure
    MRS8454 Chemical Structure
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To place orders, for customer services and technical support, please contact:

609-228-6898
[email protected] [email protected]
Find Your Local Distributor Your local distributor: Hycultec GmbHHycultec
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Top Publications Citing

Use of MCE Products

All Adenosine Receptor Isoforms

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100 mg

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  • MRS8454 Chemical Structure
    MRS8454 Chemical Structure
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  • MRS8454