1. Metabolic Enzyme/Protease
    Neuronal Signaling
  2. FAAH
  3. URB937

URB937 

Cat. No.: HY-116477
Handling Instructions

URB937 is a FAAH inhibitor and increases anandamide levels, with an IC50 of 26.8 nM. URB937 fails to affect FAAH activity in the brain.

For research use only. We do not sell to patients.

URB937 Chemical Structure

URB937 Chemical Structure

CAS No. : 1357160-72-5

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Description

URB937 is a FAAH inhibitor and increases anandamide levels, with an IC50 of 26.8 nM. URB937 fails to affect FAAH activity in the brain[1].

IC50 & Target

IC50: 26.8 nM (FAAH)[1].

In Vivo

URB937 (1 mg/kg, i.p.) administrated in mice increases anandamide levels in peripheral tissues, but not forebrain or hypothalamus[1].
URB937 (1 mg/kg, s.c.) suppresses pain responses elicited by i.p. injections of acetic acid[1].

Animal Model: Swiss Webster mice[1].
Dosage: 1 mg/kg.
Administration: S.C.
Result: Suppressesd pain responses elicited by i.p. injections of acetic acid.
Molecular Weight

354.40

Formula

C₂₀H₂₂N₂O₄

CAS No.

1357160-72-5

SMILES

O=C(OC1=CC(C2=CC=CC(C(N)=O)=C2)=C(O)C=C1)NC3CCCCC3

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

URB937URB 937URB-937FAAHFatty acid amide hydrolaseInhibitorinhibitorinhibit

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