EZH2-IN-22
EZH2-IN-22 (example 92) is a potent EZH2 inhibitor with IC50 values of <0.00051, <0.00051, 0.00052 µM for EZH2 (Y641N), EZH2 (Y641F), EZH2 (wt), respectively. EZH2-IN-22 shows antiproliferation activity.
For research use only. We do not sell to patients.
- CAS No.: 2766231-05-2
- Formula: C36H50N4O8
- Molecular Weight:666.80
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Histone Methyltransferase Isoforms
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Biological Activity
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EZH2 Y641N <0.00051 μM (IC50) |
EZH2 Y641F mutant type <0.00051 μM (IC50) |
EZH2 WT 0.00052 μM (IC50) |
Chemical Information
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CAS No. 2766231-05-2
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Molecular Weight 666.80
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Formula C36H50N4O8
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SMILES
OC(/C=C\C(O)=O)=O.CCN(C1CCOCC1)C2=C(C(C(NCC3=C(C=C(NC3=O)C)C)=O)=CC(O[C@@H]4C[C@@H](N5CCCCC5)C4)=C2)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
EZH2-IN-22 Related Classifications
HY-169958 Related Classifications
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