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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
31 Results for "
Heterocycle
" in MedChemExpress (MCE) Product Catalog:
Products (31)
31 Results for "Heterocycle" in MCE Product Catalog:
1
Target:
Thiosemicarbazide is a vitamin B6 antagonist with anti-acne activity. Thiosemicarbazide is also a well-known source in the synthesis of heterocycles, and its derivatives have potential anticancer activity. Thiosemicarbazide (TSC: HL1) reacts with metal salts, urea (U), to prepare Co(II) and Cu(I) metal complexes. Thiosemicarbazide is also used in the fields of media communications and optical storage, and in the spectrophotometric detection of metals .
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1 Cited Publications
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DuP-697 is a member of the vicinal diaryl heterocycles and a potent, irreversible, selective and orally active COX-2 inhibitor (IC50 of 10 nM and 800 nM for human COX-2 and COX-1, respectively). DuP-697 exerts antiproliferative (IC50 of 42.8 nM), antiangiogenic and apoptotic effects on HT29 colorectal cancer cells. DuP-697 inhibits prostaglandin synthesis and has anti-inflammatory, anticancer and antipyretic effects .
Cat. No.: HY-59261
CAS No.: 59489-71-3
Cat. No.: HY-W010649
CAS No.: 288-14-2
Target:
HSP Epigenetic Reader Domain ATP-binding cassette (ABC) transporters Bacterial Fungal Antibiotic
Research Areas:
Isoxazole is a member of the five-membered heterocycle drug scaffold. Isoxazole has been used as a BET bromodomain inhibitor and can improve β-cell function in a diabetic mouse model. Isoxazole and its derivatives exhibit broad biological activities (such as antimicrobial, antibacterial, antifungal, antiviral, anticancer, anti-inflammatory, immunomodulatory, analgesic, anti-tuberculosis, and anti-diabetic effects). For example, the bicyclic Isoxazole can act as an HSP90 inhibitor, and the tricyclic Isoxazole is promising as a selective multidrug resistance protein (MRP1) inhibitor .
Dehydroacetic acid sodium (Biocide 470F sodium) is a pyrone derivative. Dehydroacetic acid sodium has antibacterial, antifungal and phytotoxic activities. Dehydroacetic acid sodium can be added to cosmetics, food and beverages for preservation and other purposes. Dehydroacetic acid sodium can also be used to synthesize various heterocycles and cycloaddition products .
Dehydroacetic acid (Biocide 470F) is a pyrone derivative. Dehydroacetic acid has antibacterial, antifungal and phytotoxic activities. Dehydroacetic acid can be added to cosmetics, food and beverages for preservation and other purposes. Dehydroacetic acid can also be used to synthesize various heterocycles and cycloaddition products .
Cat. No.: HY-W002179
CAS No.: 15164-44-0
Cat. No.: HY-D1274C
Cat. No.: HY-W339545A
Cat. No.: HY-W802699
CAS No.: 1282616-74-3
Target:
Thiosemicarbazide is a vitamin B6 antagonist with anti-acne activity. Thiosemicarbazide is also a well-known source in the synthesis of heterocycles, and its derivatives have potential anticancer activity. Thiosemicarbazide (TSC: HL1) reacts with metal salts, urea (U), to prepare Co(II) and Cu(I) metal complexes. Thiosemicarbazide is also used in the fields of media communications and optical storage, and in the spectrophotometric detection of metals .
Cat. No.: HY-142048
CAS No.: 2538293-52-4
Target:
Research Areas:
BI-9466 (Compound 2) is a nuclear receptor-binding SET domain 3 (NSD3)-PWWP1 domain antagonist with a Kd of 144 µM. BI-9466 is a negative control compound of BI-9321 (HY-114208). BI-9466 has no inhibitory activity against NSD3-PWWP1 domain by introduction of a much basic nitrogen heterocycle at the 5-position of BI-9321 .
Cat. No.: HY-D1274
CAS No.: 1658416-54-6
Cat. No.: HY-D1274A
CAS No.: 2055138-89-9
Cat. No.: HY-128467R
CAS No.: 4418-26-2
Synonyms: Sodium dehydroacetate (Standard)
Target:
Research Areas:
Dehydroacetic acid sodium (Standard) (Sodium dehydroacetate (Standard)) is the analytical standard of Dehydroacetic acid sodium (HY-128467). This product is intended for research and analytical applications. Dehydroacetic acid sodium (Biocide 470F sodium) is a pyrone derivative. Dehydroacetic acid sodium has antibacterial, antifungal and phytotoxic activities. Dehydroacetic acid sodium can be added to cosmetics, food and beverages for preservation and other purposes. Dehydroacetic acid sodium can also be used to synthesize various heterocycles and cycloaddition products .
Synonyms: α-Terthiophene (Standard); α-Terthienyl (Standard); Trithiophene (Standard)
Target:
Target:
Research Areas:
Dehydroacetic acid (Standard) (Biocide 470F (Standard)) is the analytical standard of Dehydroacetic acid (HY-B1211). This product is intended for research and analytical applications. Dehydroacetic acid (Biocide 470F) is a pyrone derivative. Dehydroacetic acid has antibacterial, antifungal and phytotoxic activities. Dehydroacetic acid can be added to cosmetics, food and beverages for preservation and other purposes. Dehydroacetic acid can also be used to synthesize various heterocycles and cycloaddition products .
Cat. No.: HY-D1274B
Cat. No.: HY-149727
Target:
Research Areas:
β2AR agonist 2(compound 8a) is a β2 -Adrenergic receptor (β2AR) agonist. β2AR agonist 2 is a saturated nitrogen ring compound containing 4- to 7-membered heterocycle. β2AR agonist 2 has a chiral structure (the -R form) by carrying carbon containing the essential hydroxyl, thereby enhancing cellular glucose uptake (GU) activity and significantly stimulating glucose uptake by skeletal muscle cells. β2AR agonist 2 can be used in the study of Type 2 Diabetes (T2D) .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
