Scientific Reviews
Product Guides
Blogs
Topics
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
28 Results for "
rat PR
" in MedChemExpress (MCE) Product Catalog:
Products (28)
28 Results for "rat PR" in MCE Product Catalog:
Cat. No.: HY-106827
CAS No.: 74513-62-5
Synonyms: RU 27987
Research Areas:
Trimegestone (RU 27987) is an orally active, selective progestogen and PR ligand, with an IC50 of 7.6 nM for hPR, 4.4 nM for rabbit PR, and 3.3 nM for rat PR. Trimegestone induces Alkaline phosphatase activity. Trimegestone exhibits antiandrogenic activity (IC50 = 303 nM). Trimegestone can be used in research related to menopausal symptoms and osteoporosis .
Cat. No.: HY-123163
CAS No.: 240805-96-3
Synonyms: RWJ-66826; RTI-6617-003
Research Areas:
JNJ-1250132 (RWJ-66826) is an orally active and potent steroidal progesterone receptor (PR) antagonist, with an IC50 of 1.3 nM. JNJ-1250132 inhibits binding of the receptor to DNA in vitro. JNJ-1250132 is a potent competitive inhibitor of binding to the human glucocorticoid receptor (GR) (IC50=0.50 nM) and the rat androgen receptor (AR) (IC50=5.6 nM), and was a weak inhibitor of binding to human Estrogen receptor (ER) (IC50 >3000 nM) .
Cat. No.: HY-RS12393
Research Areas:
S1pr1 Rat Pre-designed siRNA Set A contains three designed siRNAs for S1pr1 gene (Rat), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS12396
Research Areas:
S1pr2 Rat Pre-designed siRNA Set A contains three designed siRNAs for S1pr2 gene (Rat), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS12399
Target:
Research Areas:
S1pr3 Rat Pre-designed siRNA Set A contains three designed siRNAs for S1pr3 gene (Rat), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS12402
Target:
Research Areas:
S1pr4 Rat Pre-designed siRNA Set A contains three designed siRNAs for S1pr4 gene (Rat), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS12405
Research Areas:
S1pr5 Rat Pre-designed siRNA Set A contains three designed siRNAs for S1pr5 gene (Rat), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-106827S1
Synonyms: RU 27987-13C,d3
Cat. No.: HY-108998
CAS No.: 96480-44-3
Target:
Research Areas:
Bisaramil hydrochloride is an antiarrhythmic compound with activity in inhibiting free radical generation. Bisaramil hydrochloride directly blocks sodium currents and exhibits enhanced sodium channel blocking ability. Bisaramil hydrochloride inhibits isoproterenol-induced slow calcium action potentials in cardiomyocytes. Bisaramil hydrochloride reduces heart rate and prolongs the PR, QRS, and QT intervals in the electrocardiogram, showing blocking effects on sodium and potassium channels. Bisaramil hydrochloride reduces cardiac conduction velocity, increases the threshold current for capture and atrial fibrillation, and prolongs the effective refractory period. Bisaramil hydrochloride reduces ventricular arrhythmias and eliminates mortality caused by ventricular fibrillation in ischemic rat hearts .
Cat. No.: HY-RS24725
Target:
Research Areas:
M6pr Rat Pre-designed siRNA Set A contains three designed siRNAs for M6pr gene (Rat), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-P75543
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: ACAT2; Acetoacetyl Coenzyme A Thiolase; Acetyl-CoA Acetyltransferase 2; Acetyl-Coenzyme A Acetyltransferase 2 (Acetoacetyl Coenzyme A Thiolase); Acetyl-CoA Acetyltransferase, Cytosolic; Acetyl-Coenzyme A Acetyltransferase 2; Acetyl-CoA Transferase-Like PR
Cat. No.: HY-P70233
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: KRAS; Kras-Enoph1 Fusion PRotein; PRev. KRAS2; PR310 C-K-Ras Oncogene; GTPase KRas; Small Monomeric GTPase; K-Ras4B; C-Kirsten-Ras PRotein; KRAS1; PRoto-Oncogene GTPase; V-Ki-Ras2 Kirsten rat Sarcoma 2 Viral Oncogene Homolog; KRAS-ENOPH Fusion; Kirsten Ra
Cat. No.: HY-P70233A
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: KRAS; Kras-Enoph1 Fusion PRotein; PRev. KRAS2; PR310 C-K-Ras Oncogene; GTPase KRas; Small Monomeric GTPase; K-Ras4B; C-Kirsten-Ras PRotein; KRAS1; PRoto-Oncogene GTPase; V-Ki-Ras2 Kirsten rat Sarcoma 2 Viral Oncogene Homolog; KRAS-ENOPH Fusion; Kirsten Ra
Cat. No.: HY-P704746
Purity: ≥ 90%, as determined by reducing SDS-PAGE.
Synonyms: KRAS; Kras-Enoph1 Fusion PRotein; PRev. KRAS2; PR310 C-K-Ras Oncogene; GTPase KRas; Small Monomeric GTPase; K-Ras4B; C-Kirsten-Ras PRotein; KRAS1; PRoto-Oncogene GTPase; V-Ki-Ras2 Kirsten rat Sarcoma 2 Viral Oncogene Homolog; KRAS-ENOPH Fusion; Kirsten Ra
Species:
Source:
Cat. No.: HY-P704771
Purity: ≥ 90%, as determined by reducing SDS-PAGE.
Synonyms: KRAS; Kras-Enoph1 Fusion PRotein; PRev. KRAS2; PR310 C-K-Ras Oncogene; GTPase KRas; Small Monomeric GTPase; K-Ras4B; C-Kirsten-Ras PRotein; KRAS1; PRoto-Oncogene GTPase; V-Ki-Ras2 Kirsten rat Sarcoma 2 Viral Oncogene Homolog; KRAS-ENOPH Fusion; Kirsten Ra
Cat. No.: HY-P7804
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: KRAS; Kras-Enoph1 Fusion PRotein; PRev. KRAS2; PR310 C-K-Ras Oncogene; GTPase KRas; Small Monomeric GTPase; K-Ras4B; C-Kirsten-Ras PRotein; KRAS1; PRoto-Oncogene GTPase; V-Ki-Ras2 Kirsten rat Sarcoma 2 Viral Oncogene Homolog; KRAS-ENOPH Fusion; Kirsten Ra
Cat. No.: HY-P7805
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: KRAS; Kras-Enoph1 Fusion PRotein; PRev. KRAS2; PR310 C-K-Ras Oncogene; GTPase KRas; Small Monomeric GTPase; K-Ras4B; C-Kirsten-Ras PRotein; KRAS1; PRoto-Oncogene GTPase; V-Ki-Ras2 Kirsten rat Sarcoma 2 Viral Oncogene Homolog; KRAS-ENOPH Fusion; Kirsten Ra
Cat. No.: HY-P70153
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: KRAS; Kras-Enoph1 Fusion PRotein; PRev. KRAS2; PR310 C-K-Ras Oncogene; GTPase KRas; Small Monomeric GTPase; K-Ras4B; C-Kirsten-Ras PRotein; KRAS1; PRoto-Oncogene GTPase; V-Ki-Ras2 Kirsten rat Sarcoma 2 Viral Oncogene Homolog; KRAS-ENOPH Fusion; Kirsten Ra
Cat. No.: HY-P70232
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: KRAS; Kras-Enoph1 Fusion PRotein; PRev. KRAS2; PR310 C-K-Ras Oncogene; GTPase KRas; Small Monomeric GTPase; K-Ras4B; C-Kirsten-Ras PRotein; KRAS1; PRoto-Oncogene GTPase; V-Ki-Ras2 Kirsten rat Sarcoma 2 Viral Oncogene Homolog; KRAS-ENOPH Fusion; Kirsten Ra
Cat. No.: HY-P70234
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: KRAS; Kras-Enoph1 Fusion PRotein; PRev. KRAS2; PR310 C-K-Ras Oncogene; GTPase KRas; Small Monomeric GTPase; K-Ras4B; C-Kirsten-Ras PRotein; KRAS1; PRoto-Oncogene GTPase; V-Ki-Ras2 Kirsten rat Sarcoma 2 Viral Oncogene Homolog; KRAS-ENOPH Fusion; Kirsten Ra
- 1
- 2
-
-
Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
