1. Membrane Transporter/Ion Channel
  2. Potassium Channel
  3. Pinacidil monohydrate

Pinacidil monohydrate 

Cat. No.: HY-14290A Purity: >99.0%
Handling Instructions

Pinacidil monohydrate, an antihypertensive drug, is a potassium channel activator.

For research use only. We do not sell to patients.

Pinacidil monohydrate Chemical Structure

Pinacidil monohydrate Chemical Structure

CAS No. : 85371-64-8

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 55 In-stock
Estimated Time of Arrival: December 31
5 mg USD 50 In-stock
Estimated Time of Arrival: December 31
10 mg USD 80 Get quote
25 mg USD 160 Get quote
50 mg   Get quote  
100 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

Pinacidil monohydrate, an antihypertensive drug, is a potassium channel activator.

In Vitro

Pinacidil monohydrate is a potassium channel activator[1]. Pinacidil hydrate is an antihypertensive drug of the class of agents called "potassium channel openers"[2]. Pinacidil hydrate activates the ATP-modulated potassium channels of guinea pog bladder and heart with Ki values of 104 and 251 nM, respectively[3].

Molecular Weight

263.34

Formula

C₁₃H₂₁N₅O

CAS No.

85371-64-8

SMILES

[H]O[H].CC(C)(C)C(N/C(NC#N)=N/C1=CC=NC=C1)C

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

Ethanol : 50 mg/mL (189.87 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 3.7974 mL 18.9869 mL 37.9737 mL
5 mM 0.7595 mL 3.7974 mL 7.5947 mL
10 mM 0.3797 mL 1.8987 mL 3.7974 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% EtOH    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (9.49 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% EtOH    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (9.49 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% EtOH    90% corn oil

    Solubility: ≥ 2.5 mg/mL (9.49 mM); Clear solution

*All of the co-solvents are provided by MCE.
References

Purity: >99.0%

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Product name:
Pinacidil monohydrate
Cat. No.:
HY-14290A
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