1. Neuronal Signaling
  2. AChE
  3. Rivastigmine tartrate

Rivastigmine tartrate (Synonyms: ENA 713; SDZ-ENA 713)

Cat. No.: HY-11017 Purity: 99.45%
Handling Instructions

Rivastigmine tartrate, an cholinesterase inhibitor(IC50= 5.5 uM), inhibits both butyrylcholinesterase and acetylcholinesterase IC50 value: 5.5 uM Target: AChE Rivastigmine is a parasympathomimetic or cholinergic agent for the treatment of mild to moderate dementia of the Alzheimer's type and dementia due to Parkinson's disease.

For research use only. We do not sell to patients.

Rivastigmine tartrate Chemical Structure

Rivastigmine tartrate Chemical Structure

CAS No. : 129101-54-8

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10 mM * 1 mL in Water USD 79 In-stock
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50 mg USD 72 In-stock
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200 mg USD 144 In-stock
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Description

Rivastigmine tartrate, an cholinesterase inhibitor(IC50= 5.5 uM), inhibits both butyrylcholinesterase and acetylcholinesterase IC50 value: 5.5 uM Target: AChE Rivastigmine is a parasympathomimetic or cholinergic agent for the treatment of mild to moderate dementia of the Alzheimer's type and dementia due to Parkinson's disease. The drug can be administered orally or via a transdermal patch; the latter form reduces the prevalence of side effects, which typically include nausea and vomiting. The drug is eliminated through the urine, and appears to have relatively few drug-drug interactions. Rivastigmine, a cholinesterase inhibitor, inhibits both butyrylcholinesterase and acetylcholinesterase. It is thought to work by inhibiting these cholinesterase enzymes, which would otherwise break down the brain chemical acetylcholine.

Clinical Trial
Molecular Weight

400.42

Formula

C₁₈H₂₈N₂O₈

CAS No.

129101-54-8

SMILES

O=C(OC1=CC=CC([[email protected]@H](N(C)C)C)=C1)N(CC)C.O=C(O)[[email protected]](O)[[email protected]@H](O)C(O)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

H2O : 50 mg/mL (124.87 mM; Need ultrasonic)

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Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.4974 mL 12.4869 mL 24.9738 mL
5 mM 0.4995 mL 2.4974 mL 4.9948 mL
10 mM 0.2497 mL 1.2487 mL 2.4974 mL
*Please refer to the solubility information to select the appropriate solvent.
References
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Keywords:

RivastigmineENA 713 SDZ-ENA 713ENA713ENA-713AChEAcetylcholinesteraseInhibitorinhibitorinhibit

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Product name:
Rivastigmine tartrate
Cat. No.:
HY-11017
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