1. Protein Tyrosine Kinase/RTK
  2. c-Kit

Sitravatinib (Synonyms: MGCD516; MG516)

Cat. No.: HY-16961 Purity: 99.85%
Handling Instructions

Sitravatinib?is an orally bioavailable, receptor tyrosine kinase (RTK)?inhibitor?with potential antineoplastic activity.

For research use only. We do not sell to patients.

Sitravatinib Chemical Structure

Sitravatinib Chemical Structure

CAS No. : 1123837-84-2

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply now  
10 mM * 1 mL in DMSO USD 111 In-stock
Estimated Time of Arrival: December 31
5 mg USD 80 In-stock
Estimated Time of Arrival: December 31
10 mg USD 120 In-stock
Estimated Time of Arrival: December 31
50 mg USD 300 In-stock
Estimated Time of Arrival: December 31
100 mg USD 490 In-stock
Estimated Time of Arrival: December 31
200 mg USD 820 In-stock
Estimated Time of Arrival: December 31
500 mg   Get quote  
1 g   Get quote  

* Please select Quantity before adding items.

Customer Review

  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

Sitravatinib?is an orally bioavailable, receptor tyrosine kinase (RTK)?inhibitor?with potential antineoplastic activity.

Clinical Trial
Solvent & Solubility
In Vitro: 

DMSO : ≥ 32 mg/mL (50.82 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.5881 mL 7.9405 mL 15.8811 mL
5 mM 0.3176 mL 1.5881 mL 3.1762 mL
10 mM 0.1588 mL 0.7941 mL 1.5881 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

629.68

Formula

C₃₃H₂₉F₂N₅O₄S

CAS No.

1123837-84-2

SMILES

O=C(C1(C(NC2=CC=C(F)C=C2)=O)CC1)NC3=CC=C(OC4=C5C(C=C(C6=NC=C(CNCCOC)C=C6)S5)=NC=C4)C(F)=C3

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Inquiry Information

Product Name:
Sitravatinib
Cat. No.:
HY-16961
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Sitravatinib

Cat. No.: HY-16961