USP1-IN-13
USP1-IN-13 (Compound 2) is a potent and orally active USP1 inhibitor with an IC50 value of 1.02 nM. USP1-IN-13 can be used for the study of breast cancer.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 2974433-50-4
- 分子式: C30H33F4N7O
- 分子量:583.62
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
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USP1 1.02 nM (IC50) |
USP1-IN-13 (Compound 2) (14 d) inhibits the colony-forming ability of MDA-MB-436 cells, with its IC50 value being 31.34 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
| Species | Dose | Route | Cmax | AUC0-t |
|---|---|---|---|---|
| Mice[1] | 10 mg/kg | i.g. | 1432 ng/mL | 9888 ng·h/mL |
化学情報
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CAS 番号 2974433-50-4
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分子量 583.62
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分子式 C30H33F4N7O
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SMILES
COC1=C(C(C2CC2)=NC=N1)C3=C(C4=C(C=NN4CC56CCC(CC5)(CC6)C7=NC(C(F)(F)F)=CN7C(C)C)C=N3)F
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
USP1-IN-13 関連分類
HY-176704 関連分類
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