Iso-PU-H54
Iso-PU-H54 is a purine-scaffold Grp94 inhibitor with an IC50 of 1.63 μM.
For research use only. We do not sell to patients.
- CAS No.: 852030-37-6
- Formula: C18H19N5S
- Molecular Weight:337.45
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| SK-BR-3 | IC50 |
31.8 μM
Compound: 11k
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Inhibitory concentration against SKBr3 cell line
Inhibitory concentration against SKBr3 cell line
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[PMID: 15828828] |
Iso-PU-H54 (compound 9i) inhibits recombinant Trap-1 with an IC50 of 13.8 μM and shows no significant activity against recombinant Hsp90α or Hsp90β (IC50 > 300 μM)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 852030-37-6
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Molecular Weight 337.45
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Formula C18H19N5S
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SMILES
C#CCCCN1C(=NC=2C(=NC=NC21)N)SC3=CC=C(C=C3C)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Iso-PU-H54 Related Classifications
HY-103063 Related Classifications
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