1 Result for "

CB839 derivative

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "CB839 derivative" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-114334
CAS No.: 2247127-79-1
Purity:  98.09%
Synonyms: CB839 derivative
Target:  

Glutaminase

Research Areas:  

Cancer

Glutaminase-IN-1 (CB839 derivative), a CB839 derivative, is an allosteric inhibitor of 1,3,4-selenadiazole-containing kidney-type glutaminase (KGA), with an IC50 of 1 nM. Glutaminase-IN-1 (CB839 derivative) shows improved cellular uptake and antitumor activity.
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