1 Result for "

Fedratinib-d9

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "Fedratinib-d9" in MCE Product Catalog:

Cat. No.: HY-10409S
Synonyms: TG-101348-d9; SAR 302503-d9
Fedratinib-d9 (TG-101348-d9) is deuterium labeled Fedratinib. Fedratinib (TG-101348) is a potent, selective, ATP-competitive and orally active JAK2 inhibitor with IC50s of 3 nM for both JAK2 and JAK2V617F kinase. Fedratinib shows 35- and 334-fold selectivity over JAK1 and JAK3, respectively. Fedratinib induces cancer cell apoptosis and has the potential for myeloproliferative disorders research .
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