1. GPCR/G Protein
  2. Adenosine Receptor
  3. FSCPX

FSCPX 

Cat. No.: HY-116042
Handling Instructions

FSCPX is a potent and selective irreversible antagonist of A1 adenosine receptor (A1AR), with low nanomolar potency for binding to the A1AR. FSCPX could modifies the effect of NBTI, a nucleoside transport inhibitor, by reducing the interstitial adenosine level in the guinea pig atrium.

For research use only. We do not sell to patients.

FSCPX Chemical Structure

FSCPX Chemical Structure

CAS No. : 156547-56-7

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Description

FSCPX is a potent and selective irreversible antagonist of A1 adenosine receptor (A1AR), with low nanomolar potency for binding to the A1AR. FSCPX could modifies the effect of NBTI, a nucleoside transport inhibitor, by reducing the interstitial adenosine level in the guinea pig atrium[1][2].

IC50 & Target

A1AR[1]

In Vitro

FSCPX irreversibly blocks the binding of [3H]-8-cyclopentyl-1,3dipropylxanthine ([3H]DPCPX), with an IC50 of 11.8±3.2 nM in DDT1 MF2 cells[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

506.55

Formula

C₂₃H₂₇FN₄O₆S

CAS No.

156547-56-7

SMILES

O=C(OCCCN(C(N1CCC)=O)C2=C(N=C(C3CCCC3)N2)C1=O)C4=CC=C(S(=O)(F)=O)C=C4

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

FSCPXAdenosine ReceptorP1 receptorirreversibleA1adenosineA1ARNBTIdenosineInhibitorinhibitorinhibit

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