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2841308-96-9

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1 Results for "2841308-96-9" in MCE Product Catalog:

Cat. No.: HY-162412
CAS No.: 2841308-96-9
Research Areas:  

Cancer

PROTAC AR/AR-V7 degrader-1 (27c) is a PROTAC-based and dual AR, AR-V7 degrader, with DC50 values of 2.67 and 2.64 μM for AR and AR-V7, respectively. PROTAC AR/AR-V7 degrader-1 (27c) induces apoptosis (Red: AR antagonist; Blue: E3 ligase ligand; Black: linker) .
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