1 Result for "

3066972-97-9

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "3066972-97-9" in MCE Product Catalog:

Cat. No.: HY-170366
CAS No.: 3066972-97-9
Target:  

VEGFR Apoptosis

Research Areas:  

Cancer

VEGFR-2-IN-58 (Compound 7b) inhibits VEGFR-2 with an IC50 of 42.5 nM. VEGFR-2-IN-58 displays selective cytotoxicity against cancer cells. VEGFR-2-IN-58 shows cellular growth arrest at the G2/M phase in cancer cells. VEGFR-2-IN-58 induces cancer cells Apoptosis, increasing BAX expression and reducing Bcl2 expression. VEGFR-2-IN-58 inhibits wound closure in cancer cells .
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