1 Result for "

317844-33-0

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "317844-33-0" in MCE Product Catalog:

Cat. No.: HY-19858
CAS No.: 317844-33-0
Target:  

iGluR

Research Areas:  

Neurological Disease

LY-466195 is a selective and competitive GLUK5 receptor antagonist. LY-466195 antagonizes Kainate-induced currents with an IC50 value of 0.045 μM in rat dorsal root ganglion neurons. In HEK293 cells transfected with GLUK5, GLUK2/GLUK5, or GLUK5/GLUK66 receptors, LY466195 produces IC50 values of 0.08 μM, 0.34 μM, and 0.07 μM, respectively .
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