1 Result for "

3D53 monoacetate

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "3D53 monoacetate" in MCE Product Catalog:

Cat. No.: HY-106178D
CAS No.: 852629-88-0
Synonyms: 3D53 monoacetate
Target:  

Endogenous Metabolite

Research Areas:  

Inflammation/Immunology

PMX 53 monoacetate (3D53 monoacetate) is a potent orally active CD88 (C5aR) antagonist that inhibits C5a-induced neutrophil myeloperoxide release and chemotactic activity. PMX 53 monoacetate has an IC50 value of 20 nM against C5a-induced neutrophil myeloperoxide release. >The value is 22 nM, and the IC50 value of the chemotactic activity is 75 nM. PMX 53 monoacetate is also an agonist of MrgX2 .
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