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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
4 Results for "
CB2R antagonist 4
" in MedChemExpress (MCE) Product Catalog:
Products (4)
4 Results for "CB2R antagonist 4" in MCE Product Catalog:
Cat. No.: HY-175784
CAS No.: 1341021-90-6
Target:
Research Areas:
CB2R antagonist 4 is a selective CB2R antagonist/inverse agonist with a pKi of 6.54. CB2R antagonist 4 shows a ≥11-fold selectivity towards CB2R over CB1R and can be utilized in neurological research .
Cat. No.: HY-174846
Research Areas:
TRPM8 antagonist 4 prodrug (Compound 8b) is an orally active CB2R agonist (EC50: 51.2 nM) and a weak TRPM8 antagonist. TRPM8 antagonist 4 prodrug is a prodrug of TRPM8 antagonist 4 (HY-174825). TRPM8 antagonist 4 prodrug exhibits anti-inflammatory and analgesic activities and can be used in the research of inflammation-related pain disorders .
Cat. No.: HY-174825
CAS No.: 3107363-68-5
Cat. No.: HY-155481A
Target:
Research Areas:
CB2 receptor antagonist 4 (compound (R)-1) is a CB2R-selective inverse agonist with a Kd value of 39 nM .
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Protocols
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