TRPM8 antagonist 4 prodrug
TRPM8 antagonist 4 prodrug (Compound 8b) is an orally active CB2R agonist (EC50: 51.2 nM) and a weak TRPM8 antagonist. TRPM8 antagonist 4 prodrug is a prodrug of TRPM8 antagonist 4 (HY-174825). TRPM8 antagonist 4 prodrug exhibits anti-inflammatory and analgesic activities and can be used in the research of inflammation-related pain disorders.
For research use only. We do not sell to patients.
- Formula: C22H29NO4
- Molecular Weight:371.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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CB2 51.2 nM (IC50) |
TRPM8 |
Chemical Information
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Molecular Weight 371.47
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Formula C22H29NO4
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SMILES
C/C(C)=C/CC/C(C)=C/COC1=CC(C2CC2)=C(C(N)=O)C(OC(C)=O)=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
TRPM8 antagonist 4 prodrug Related Classifications
HY-174846 Related Classifications
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