2 Results for "

non-REM sleep

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "non-REM sleep" in MCE Product Catalog:

Cat. No.: HY-106547
CAS No.: 99593-25-6
Target:  

GABA Receptor

Research Areas:  

Neurological Disease

Rilmazafone (450191S) is an orally active sleep inducer. Rilmazafone targets cytochrome P-450b and cytochrome P-450e. Rilmazafone induces hepatic drug-metabolizing enzyme activity in rats, mice and dogs. Rilmazafone is applicable for insomnia-related research .
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Cat. No.: HY-184060
CAS No.: 1704716-36-8
Target:  

GABA Receptor

Research Areas:  

Neurological Disease

ASP8062 is an orally active, blood-brain barrier-permeable selective GABAB receptor positive allosteric modulator. ASP8062 enhances GABA-mediated activation of GABAB receptors and strengthens GABAergic neurotransmission. ASP8062 reverses Reserpine (HY-N0480)-induced myalgia, regulates the sleep-wake cycle, increases delta wave power during non-REM sleep, and impairs motor coordination at high doses. ASP8062 penetrates the central nervous system with a half-life of 40-50 h. ASP8062 can be used in research related to opioid use disorder, fibromyalgia, chronic pain, and alcohol use disorder .
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