CTR/AMYR agonist-2
CTR/AMYR agonist-2 is a fused heterocyclic amide/sulfonamide compound, as well as a calcitonin G protein-coupled receptor (CGRP Receptor) / amylin receptor agonist. CTR/AMYR agonist-2 shows potential for application in research related to diseases such as obesity and type 2 diabetes.
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- Formel: C36H35F2N7O6
- Molecular Weight:699.70
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
Beschreibung
In Vitro
CTR/AMYR agonist-2 (Example 117) exhibits a geometric mean EC50 of 1.89 nM and an asymptotic maximum response of 128% in the HTRF‑cAMP agonism functional assay using CHO cells expressing human calcitonin receptor[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Molecular Weight 699.70
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Formel C36H35F2N7O6
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SMILES
O[C@@H](C1)[C@@H](NC(C2=COC(C3=C(C4=NN=C(CN(C)C)O4)C(CCC5=CC=C(F)C=C5)=NC(O[C@H](C)[C@@H](C)N6)=C3C6=O)=N2)=O)C7=C1C=C(F)C=C7
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)