2. GPCR/G Protein Neuronal Signaling
  3. Dopamine Receptor Vasopressin Receptor Adrenergic Receptor
  4. Docarpamine

Docarpamine is an orally active dopamine prodrug that can be hydroxylated in the small intestine and liver to form active dopamine. Docarpamine mainly activates D1-like receptors in peripheral blood vessels to lower blood pressure and heart rate in a state of spontaneous hypertension. Docarpamine exerts a pressor and tachycardic effect by activating D1-like receptors, vasopressin V1 receptors, and α-adrenergic receptors in normal blood pressure conditions. Docarpamine can be used for research on renal vascular dilation and diuresis.

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Docarpamine

Docarpamine Chemical Structure

CAS No. : 74639-40-0

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Docarpamine Related Antibodies

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Dopamine Receptor D1 Receptor D2 Receptor D3 Receptor D4 Receptor D5 Receptor

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V1a Receptor  V1b Receptor  V2 Receptor 

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α adrenergic receptor β adrenergic receptor

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Description

Docarpamine is an orally active dopamine prodrug that can be hydroxylated in the small intestine and liver to form active dopamine. Docarpamine mainly activates D1-like receptors in peripheral blood vessels to lower blood pressure and heart rate in a state of spontaneous hypertension. Docarpamine exerts a pressor and tachycardic effect by activating D1-like receptors, vasopressin V1 receptors, and α-adrenergic receptors in normal blood pressure conditions. Docarpamine can be used for research on renal vascular dilation and diuresis[1][2].

IC50 & Target[1]

D1 Receptor

 

α adrenergic receptor

 

Molecular Weight

470.54

Formula

C21H30N2O8S
CAS No.
SMILES

CCOC(OC1=C(C=C(C=C1)CCNC([C@@H](NC(C)=O)CCSC)=O)OC(OCC)=O)=O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Docarpamine Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Docarpamine74639-40-0Dopamine ReceptorVasopressin ReceptorAdrenergic ReceptorBeta Receptordopamine prodrugmean arterial pressureheart ratespontaneously hypertensive rats (SHR)Wistar-Kyoto rats (WKY)D1-like receptorsSCH 23390alpha-adrenergic receptorsvasopressin V1 receptorsInhibitorinhibitorinhibit

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