GW694481
Based on 1 publication(s) in Google Scholar
GW694481 is an ApoA1 upregulator with IC50 values of 2.1 μM for CYP2C9 inhibition and 17.0 μM for CYP3A4 inhibition. GW694481 upregulates ApoA1 expression in human hepatic cells.GW694481 can be used for the research of atherosclerosis.
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- No. CAS: 1373353-95-7
- Fòrmula: C21H18N4O2
- Peso molecular:358.39
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Publications Citing Use of MedChemExpress (MCE) GW694481
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Actividad biológica
GW694481 upregulates ApoA1 expression in stably transfected HepG2 cells with an EC170 of 0.52 μM, and inhibits CYP 2C9 and CYP 3A4 with IC50 values of 2.1 μM and 17.0 μM, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 1373353-95-7
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Peso molecular 358.39
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Fòrmula C21H18N4O2
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SMILES
O=C(C1=CN=C2C=C(C3=C(C)ON=C3C)C=CC2=C1NC4=CC=CC=C4)N
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications (1)
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Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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