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Cat. No.: HY-162892

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BRD4-IN-9

BRD4-IN-9 is an orally active BRD4 inhibitor with an IC₅₀ value of 9.4 nM. BRD4-IN-9 can suppress tumor growth in a mouse melanoma xenograft model.

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CAS No.: 2468959-08-0
화학식: C₂₄H₂₃N₃O₃
분자량:401.46

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (267 KB)

BRD4-IN-9 Chemical Structure

CAS No.: 2468959-08-0

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

제품 설명

BRD4-IN-9 is an orally active BRD4 inhibitor with an IC₅₀ value of 9.4 nM. BRD4-IN-9 can suppress tumor growth in a mouse melanoma xenograft model^[1].

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Chemical Information

CAS No. 2468959-08-0
분자량 401.46
화학식 C₂₄H₂₃N₃O₃
SMILES

CN(C(C=C1)=O)C=C1C2=CC=C(N=C(C3CCOCC3)N4)C4=C2OC5=CC=CC=C5
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (267 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Horai Y, et al. A novel 7-phenoxy-benzimidazole derivative as a potent and orally available BRD4 inhibitor for the treatment of melanoma. Bioorg Med Chem. 2024 Oct 1;112:117882. [Content Brief]

Calculators

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
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BRD4-IN-9

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Biological Activity

Chemical Information

순도&문서

References

Calculators

Help & FAQs

BRD4-IN-9 Related Classifications

HY-162892 Related Classifications