10 Results for "

Acepromazine

" in MedChemExpress (MCE) Product Catalog:
Products (10)

10 Results for "Acepromazine" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-B1506
CAS No.: 61-00-7
Synonyms: Acetopromazine; Acetylpromazine
Target:  

Adrenergic Receptor

Research Areas:  

Neurological Disease

Acepromazine (Acetopromazine) is a phenothiazine tranquilizer and is alpha-adrenoceptor antagonist .
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1
1 Cited Publications
Cat. No.: HY-B1506A
CAS No.: 3598-37-6
Synonyms: Acetopromazine maleate; Acetylpromazine maleate
Target:  

Adrenergic Receptor

Research Areas:  

Neurological Disease

Acepromazine (Acetopromazine) maleate is a phenothiazine tranquilizer and is alpha-adrenoceptor antagonist .
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Cat. No.: HY-169357
Research Areas:  

Cancer

Acepromazine-1-piperazinepropanamine (compound 10) is a synthesized E3 ligase ligand-linker conjugate (E3 Ligase Ligand-Linker Conjugate) that incorporates a TRIM21 ligand and a linker. Acepromazine-1-piperazinepropanamine can be connected to the target protein ligand to form a PROTAC molecule, TrimTAC1 (HY-169355) .
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Cat. No.: HY-169325
Research Areas:  

Cancer

(S)-ACE‑OH is the active metabolite of Acepromazine (HY-B1506), acting as a molecular glue degrader. (S)-ACE-OH induces functional interaction between TRIM21 and NUP98, promoting protein ubiquitination and degradation of TRIM21 at the nuclear pore complex. (S)-ACE-OH triggers nucleocytoplasmic transport disorder and exerts interferon-potentiated cytotoxic effects on certain cancer cells. (S)-ACE-OH can be used in cancer-related research .
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Cat. No.: HY-169357B
Research Areas:  

Cancer

Acepromazine-1-piperazinepropanamine dihydrochloride (compound 10) is a synthesized E3 ligase ligand-linker conjugate (E3 Ligase Ligand-Linker Conjugate) that incorporates a TRIM21 ligand and a linker. Acepromazine-1-piperazinepropanamine dihydrochloride can be connected to the target protein ligand to form a PROTAC molecule, TrimTAC1 (HY-169355) .
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Cat. No.: HY-169356
CAS No.: 102951-20-2
Target:  

Ligands for E3 Ligase

Research Areas:  

Cancer

Acepromazine-OTs is a TRIM21 ligand used in the recruitment of the TRIM21 protein. Acepromazine-OTs can be connected to the target protein ligand through a linker to form a PROTAC molecule, TrimTAC1 (HY-169355) .
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Cat. No.: HY-B1506AR
CAS No.: 3598-37-6
Synonyms: Acetopromazine maleate (Standard); Acetylpromazine maleate (Standard)
Acepromazine (maleate) (Standard) is the analytical standard of Acepromazine (maleate). This product is intended for research and analytical applications. Acepromazine (Acetopromazine) maleate is a phenothiazine tranquilizer and is alpha-adrenoceptor antagonist.
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Cat. No.: HY-B1506AS
CAS No.: 1331655-50-5
Synonyms: Acetopromazine-d6 maleate; Acetylpromazine-d6 maleate
Acepromazine-d6 (maleate) (Acetopromazine-d6 (maleate)) is deuterium labeled Acepromazine (maleate). Acepromazine (Acetopromazine) maleate is a phenothiazine tranquilizer and is alpha-adrenoceptor antagonist .
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Cat. No.: HY-W774927S
CAS No.: 1173022-70-2
Acepromazine-d6 hydrochloride is the deuterium labeled Acepromazine hydrochloride. Acepromazine (Acetopromazine) is a phenothiazine tranquilizeran and alpha-adrenoceptor antagonist .
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Cat. No.: HY-175948
CAS No.: 3033297-50-3
Research Areas:  

Others

Lenalidomide-CO-C3-NH-alkynes is an E3 ligase ligand-linker conjugate comprising Lenalidomide (HY-A0003) and a linker. Acepromazine-1-piperazinepropanamine dihydrochloride can be conjugated to a target protein ligand to form a PROTAC molecule—for instance, the PROTAC EGFR degrader 7 (HY-147858) .
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