3 Results for "

GRPR antagonist 1

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "GRPR antagonist 1" in MCE Product Catalog:

Cat. No.: HY-115974
CAS No.: 3052544-28-9
Target:  

Bombesin Receptor

Research Areas:  

Cancer

GRPR antagonist-1 is a potent gastrin releasing peptide receptor (GRPR) antagonist, having the cytotoxicity against certain cancer cells (IC50 of 4.97, 4.36 and 3.40 μM in PC3, Pan02 and HGC-27 cells, respectively). GRPR antagonist-1 inhibits HGC-27 cell viability by decreasing the Bcl-2 level and increasing the Bax level, causing apoptosis, with anticancer activity .
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1
1 Cited Publications
Cat. No.: HY-P0107A
CAS No.: 1217463-61-0
Target:  

Bombesin Receptor

Research Areas:  

Inflammation/Immunology

RC-3095 TFA is a selective bombesin/gastrin releasing peptide receptor (GRPR) antagonist . RC-3095 TFA exerts protective effects by reducing gastric oxidative injury in the arthritic mice .
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1
1 Cited Publications
Cat. No.: HY-P0107
CAS No.: 138147-78-1
Target:  

Bombesin Receptor

Research Areas:  

Inflammation/Immunology

RC-3095 is a bombesin/gastrin releasing peptide receptor (GRPR) antagonist . RC-3095 exerts protective effects by reducing gastric oxidative injury in the arthritic mice .
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