11 Results for "

KISS1R

" in MedChemExpress (MCE) Product Catalog:
Products (11)

11 Results for "KISS1R" in MCE Product Catalog:

4
4 Cited Publications
Cat. No.: HY-P2161B
Target:  

Kisspeptin Receptor

Research Areas:  

Cancer

TAK-683 acetate is a potent full KISS1 receptor (KISS1R) agonist (IC50=170 pM) with improved metabolic stability. TAK-683 acetate is a nonapeptide metastin analog, exhibits agonistic activities to KISS1R with EC50 values of 0.96 nM and 1.6 nM for human and rat, respectively [1]. TAK-683 acetate depletes GnRH in the hypothalamus and reduces plasma FSH, LH, and testosterone levels in vivo, it has the potential for the study of hormone-dependent prostate cancer [1] .
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3
3 Cited Publications
Cat. No.: HY-P0076
CAS No.: 1234319-68-6
Synonyms: MVT-602
Target:  

Kisspeptin Receptor

Research Areas:  

Cancer

TAK-448 (MVT-602) is a potent and full KISS1R agonist with an IC50 of 460 pM and an EC50 of 632 pM [1].
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3
3 Cited Publications
Cat. No.: HY-P0076A
CAS No.: 1470374-22-1
Synonyms: MVT-602 acetate
Target:  

Kisspeptin Receptor

Research Areas:  

Cancer

TAK-448 acetate (MVT-602 acetate) is a potent and full KISS1R agonist with an IC50 of 460 pM and an EC50 of 632 pM [1].
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Cat. No.: HY-RS07316
Research Areas:  

Others

KISS1R Human Pre-designed siRNA Set A contains three designed siRNAs for KISS1R gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.

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Cat. No.: HY-P10489
CAS No.: 374675-19-1
Target:  

Kisspeptin Receptor

Research Areas:  

Cancer

Kisspeptin-14 human is a peptide hormone encoded by the KiSS-1 gene. Kisspeptin-14 human, along with several other similar peptide hormones, is produced from a common precursor protein by cleavage by different proteases. Kisspeptin-14 human is an endogenous ligand of KISS1R. Kisspeptin-14 human has the same receptor binding efficiency and potency as full-length kisspeptin. Kisspeptin-14 human binds to its receptor GPR54 and is able to activate this G protein-coupled receptor and activate multiple intracellular signaling pathways. Kisspeptin-14 human can be used to study reproductive development and tumor metastasis [1].
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Cat. No.: HY-RS07317
Research Areas:  

Others

Kiss1r Mouse Pre-designed siRNA Set A contains three designed siRNAs for Kiss1r gene (Mouse), as well as a negative control, a positive control, and a FAM-labeled negative control.

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Cat. No.: HY-RS07318
Research Areas:  

Others

Kiss1r Rat Pre-designed siRNA Set A contains three designed siRNAs for Kiss1r gene (Rat), as well as a negative control, a positive control, and a FAM-labeled negative control.

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Cat. No.: HY-P2161
CAS No.: 872719-49-8
Target:  

Kisspeptin Receptor

Research Areas:  

Cancer

TAK-683 is a potent full KISS1 receptor (KISS1R) agonist (IC50=170 pM) with improved metabolic stability. TAK-683 is a nonapeptide metastin analog, exhibits agonistic activities to KISS1R with EC50 values of 0.96 nM and 1.6 nM for human and rat, respectively [1]. TAK-683 depletes GnRH in the hypothalamus and reduces plasma FSH, LH, and testosterone levels in vivo, it has the potential for the study of hormone-dependent prostate cancer [1] .
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Cat. No.: HY-P2191
CAS No.: 872717-97-0
Target:  

Kisspeptin Receptor

Research Areas:  

Endocrinology

KISS1-305, the Metastin/Kisspeptin analog, is a prototype peptide and a chemical probe. KISS1-305 has suboptimal KISS1R agonistic activity, and resists plasma protease degradation [1].
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Cat. No.: HY-P2161A
Target:  

Kisspeptin Receptor

Research Areas:  

Cancer

TAK-683 TFA is a potent full KISS1 receptor (KISS1R) agonist (IC50=170 pM) with improved metabolic stability. TAK-683 TFA is a nonapeptide metastin analog, exhibits agonistic activities to KISS1R with EC50 values of 0.96 nM and 1.6 nM for human and rat, respectively [1]. TAK-683 TFA depletes GnRH in the hypothalamus and reduces plasma FSH, LH, and testosterone levels in vivo, it has the potential for the study of hormone-dependent prostate cancer [1] .
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Cat. No.: HY-P810743
Synonyms: AXOR12, GPR54, KISS1R, KISS-1 receptor, KISS-1R, G-protein coupled receptor 54, G-protein coupled receptor OT7T175, Hypogonadotropin-1, KISSpeptins receptor, Metastin receptor, hOT7T175

Host:  

Rabbit

Application:  

WB

Reactivity:  

Human, Mouse, Rat

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