1 Result for "

MD220661

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "MD220661" in MCE Product Catalog:

Cat. No.: HY-124885
CAS No.: 73423-35-5
Target:  

Monoamine Oxidase VAP-1

Research Areas:  

Metabolic Disease

MD 220661 is a semicarbazide-sensitive amine oxidase (SSAO) and monoamine oxidase (MAO) inhibitor, and serves as a major metabolite of MD 240928 in rat brain. MD 220661 acts as a substrate for SSAO and exhibits reversible, selective MAO-B inhibition in rat tissues; in the absence of semicarbazide, its inhibitory potency against MAO-A activity decreases with prolonged pre-incubation time. MD 220661 is applicable to studies related to enzyme-catalyzed metabolism .
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