8 Results for "

UK88525

" in MedChemExpress (MCE) Product Catalog:
Products (8)

8 Results for "UK88525" in MCE Product Catalog:

8
8 Publications Verification
Cat. No.: HY-A0033
CAS No.: 133099-04-4
Synonyms: UK-88525
Darifenacin (UK-88525) is a selective and orally active M3 muscarinic receptor (M3R) antagonist with a pKi of 8.9. Darifenacin binds >20-fold more specifically to M3R than to other muscarinic receptors. Darifenacin can be used in the study of urinary incontinence and other symptoms of overactive bladder. Darifenacin inhibits tumor growth in colorectal cancer cells and has anti-tumor effects .
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8
8 Publications Verification
Cat. No.: HY-A0012
CAS No.: 133099-07-7
Synonyms: UK-88525 hydrobromide
Darifenacin (UK-88525) hydrobromide is a selective and orally active M3 muscarinic receptor (M3R) antagonist with a pKi of 8.9. Darifenacin hydrobromide binds >20-fold more specifically to M3R than to other muscarinic receptors. Darifenacin hydrobromide can be used in the study of urinary incontinence and other symptoms of overactive bladder. Darifenacin hydrobromide inhibits tumor growth in colorectal cancer cells and has anti-tumor effects .
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1
1 Cited Publications
Cat. No.: HY-22437
CAS No.: 133033-93-9
Synonyms: (±)-UK-88525
Target:  

mAChR

Research Areas:  

Neurological Disease Cancer

(±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective M3 muscarinic receptor antagonist .
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Cat. No.: HY-A0033S1
CAS No.: 1095598-84-7
Synonyms: UK-88525-d4
Darifenacin-d4 is the deuterium labeled Darifenacin . Darifenacin(UK88525) is a selective M3 muscarinic receptor antagonist with pKi of 8.9. IC50 value: 8.9 (pKi) .
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Cat. No.: HY-A0012R
CAS No.: 133099-07-7
Synonyms: UK-88525 hydrobromide (Standard)
Darifenacin (hydrobromide) (Standard) is the analytical standard of Darifenacin (hydrobromide). This product is intended for research and analytical applications. Darifenacin (hydrobromide) is a selective and orally active M3 muscarinic receptor (M3R) antagonist with a pKi of 8.9. Darifenacin (hydrobromide) binds >20-fold more specifically to M3R than to other muscarinic receptors. Darifenacin (hydrobromide) can be used in the study of urinary incontinence and other symptoms of overactive bladder. Darifenacin (hydrobromide) inhibits tumor growth in colorectal cancer cells and has anti-tumor effects .
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Cat. No.: HY-W746075A
CAS No.: 2416229-88-2
Target:  

mAChR

Research Areas:  

Neurological Disease

(±)-Darifenacin N-Oxide is the impurity of Darifenacin (HY-A0033). Darifenacin (UK-88525) is a selective and orally active M3 muscarinic receptor (M3R) antagonist with a pKi of 8.9 .
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Cat. No.: HY-22437S
CAS No.: 1189701-43-6
Synonyms: (±)-UK-88525-d4
(±)-Darifenacin-d4 is deuterium labeled (±)-Darifenacin. (±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective M3 muscarinic receptor antagonist .
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Cat. No.: HY-22437S1
CAS No.: 2747914-16-3
Synonyms: (±)-UK-88525-d4 hydrobromide
(±)-Darifenacin-d4 (hydrobromide) is deuterium labeled (±)-Darifenacin. (±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective M3 muscarinic receptor antagonist[1].
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