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Results for "

narcotic

" in MedChemExpress (MCE) Product Catalog:

By Targets:	5-HT Receptor (1) Acyltransferase (2) AMPK (1) Biochemical Assay Reagents (1) Calcium Channel (2) COX (2) Dopamine Receptor (1) Drug Derivative (1) GABA Receptor (1) Insecticide (1) Isotope-Labeled Compounds (1) Mucin (1) Potassium Channel (5) Reference Standards (3) Sodium Channel (5) UGT (1)
By Research Areas:	Cancer (2) Cardiovascular Disease (2) Infection (1) Inflammation/Immunology (7) Metabolic Disease (3) Neurological Disease (21)

Inhibitors & Agonists

Natural
Products

Isotope-Labeled Compounds

Cat. No.	Product Name	Target	Research Areas	Chemical Structure

HY-B0264

Guaifenesin Guaiacol glyceryl ether; Guaiphenesin; Glycerol guaiacolate	Mucin	Neurological Disease Inflammation/Immunology
Guaifenesin (Guaiacol glyceryl ether), a constituent of guaiac resin from the wood of Guajacum officinale Linné, is an expectorant. Guaifenesin can alleviate cough discomfortby increasing sputum volume and decreasing its viscosity, thereby promoting effective cough .

HY-B1551

Benzonatate Benzononatine	Sodium Channel	Neurological Disease
Benzonatate (Benzononatine) is an orally active and non-narcotic peripheral antitussive agent. Benzonatate is a reversible voltage-gated Na ⁺ channels inhibitor. Benzonatate dampens the activity of cough stretch receptors .

HY-B1430

Butamben Butyl 4-aminobenzoate	Calcium Channel Sodium Channel Potassium Channel	Neurological Disease
Butamben (Butyl 4-aminobenzoate) results in long-lasting relief from pain, without impairing motor function or other sensory functions .

HY-121685A

Tipepidine hydrochloride 1 Publications Verification	Potassium Channel	Neurological Disease
Tipepidine hydrochloride reversibly inhibits dopamine (DA) D₂ receptor-mediated GIRK currents (I_DA(GIRK)) with an IC₅₀ of 7.0 μM. Tipepidine hydrochloride subsequently activates VTA dopamine neuron . Tipepidine hydrochloride, a non-narcotic antitussive, exerts an antidepressant-like effect .

HY-103479

GOAT-IN-1	Acyltransferase	Cardiovascular Disease Neurological Disease Metabolic Disease Cancer
GOAT-IN-1 is an inhibitor of ghrelin O-acyltransferase (GOAT), which could be useful for the prophylaxis or treatment of obesity, diabetes, hyperlipidemia, metabolic, non-alcoholic fatty liver, steatohepatitis, sarcopenia, appetite control, alcohol/narcotic dependence, Alzheimer’s disease, Parkinson’s disease, cerebrovascular dementia, cerebral apoplexy, cerebral infarction, cardic disease, some kind of tumors.

HY-A0235

Antrafenine Stakane	COX	Neurological Disease
Antrafenine (Stakane) is a non-narcotic analgesic. Antrafenine demonstrates central analgesic effects in acetic acid writhing test and mouse hot plate test experiments. Antrafenine significantly alleviates the pain of osteoarthritis. Antrafenine exhibits mild anti-inflammatory activity in a rat toe edema model. Antrafenine can be used in pain and anti-inflammatory research .

HY-133024

Flumexadol	5-HT Receptor	Neurological Disease
Flumexadol is a selective and affinity 5-HT_2C receptor agonist with a K_i of 25 nM for the (+)-enantiomer of Flumexadol, and is 40-fold selective over the 5-HT_2A receptor. Flumexadol is an orally active non-narcotic analgesic .

HY-W748379

Fenyramidol (±)-Phenyramidol	Drug Derivative	Neurological Disease
Fenyramidol is an Aminopyridine derivative. Fenyramidol can be used as a moderately potent, non-narcotic muscle relaxant with concomitant analgesic activity .

HY-136653

Ciramadol WY 15705	UGT	Neurological Disease
Ciramadol (WY 15705) is a potent and orally active analgesic agent with both narcotic agonist and UDP-glucuronyltransferase modulator properties . Ciramadol (WY 15705) can be used for postoperative pain research research.

HY-121685

Tipepidine	Potassium Channel	Neurological Disease
Tipepidine reversibly inhibits dopamine (DA) D₂ receptor-mediated GIRK currents (I_DA(GIRK)) with an IC₅₀ of 7.0 μM. Tipepidine subsequently activates VTA dopamine neuron . Tipepidine, a non-narcotic antitussive, exerts an antidepressant-like effect .

HY-119912

Antrafenine dihydrochloride Stakane dihydrochloride	COX	Neurological Disease Inflammation/Immunology
Antrafenine (Stakane) dihydrochloride is a non-narcotic analgesic. Antrafenine dihydrochloride demonstrates central analgesic effects in acetic acid writhing test and mouse hot plate test experiments. Antrafenine dihydrochloride significantly alleviates osteoarthritis pain. Antrafenine dihydrochloride exhibits mild anti-inflammatory activity in a rat toe edema model. Antrafenine dihydrochloride can be used for pain and anti-inflammatory research .

HY-122216

LY 88329	Biochemical Assay Reagents	Neurological Disease
LY 88329 is a potent narcotic antagonist .

HY-105733A

Suxemerid disulfate	Others	Others
Suxemerid disulfate is a non-narcotic cough suppressant .

HY-100294

Ruzadolane UP 26-91	Others	Neurological Disease
Ruzadolane (UP 26-91) is a non-narcotic, centrally-acting analgesic agent.

HY-B1430R

Butamben (Standard) Butyl 4-aminobenzoate (Standard)	Reference Standards Calcium Channel Sodium Channel Potassium Channel	Neurological Disease
Butamben (Standard) is the analytical standard of Butamben. This product is intended for research and analytical applications. Butamben (Butyl 4-aminobenzoate) results in long-lasting relief from pain, without impairing motor function or other sensory functions .

HY-128418

Benzonatate (PEGn)	Sodium Channel	Neurological Disease Inflammation/Immunology
Benzonatate (PEGn) is a unique non-narcotic antitussive agent that has sodium channel-blocking properties and anesthetic effects on the respiratory stretch receptors .

HY-156061

NAP-1	GABA Receptor	Neurological Disease Inflammation/Immunology
NAP-1 is a compound with agent that can suppress or relieve pain. effects. NAP-1 enhances the inhibitory current by binding to a specific site of GABAaR, resulting in a narcotic effect. NAP-1 can be used in research to develop clinical agent that can suppress or relieve pain .

HY-B1551R

Benzonatate (Standard) Benzononatine (Standard)	Reference Standards Sodium Channel	Neurological Disease
Benzonatate (Standard) (Benzononatine (Standard)) is the analytical standard of Benzonatate (HY-B155). This product is intended for research and analytical applications. Benzonatate (Benzononatine) is an orally active and non-narcotic peripheral antitussive agent. Benzonatate is a reversible voltage-gated Na ⁺ channels inhibitor. Benzonatate dampens the activity of cough stretch receptors.

HY-B0264S1

Guaifenesin-d5	Isotope-Labeled Compounds	Neurological Disease Inflammation/Immunology
Guaifenesin-d₅ is the deuterium labeled Guaifenesin. Guaifenesin (Guaiacol glyceryl ether), a constituent of guaiac resin from the wood of Guajacum officinale Linné, is an expectorant. Guaifenesin can alleviate cough discomfortby increasing sputum volume and decreasing its viscosity, thereby promoting effective cough. Guaifenesin also has narcotic effect .

HY-N7869

Celangulin VII	Insecticide	Infection
Celangulin VII is a β-dihydroagarofuran sesquiterpene polyol ester present in the root bark of Celastrus angulatus. Celangulin VII exhibits insecticidal and narcotic activities against the 4th-instar larvae of Mythimna separata. Celangulin VII can be used in insecticide-related research .

HY-103479R

GOAT-IN-1 (Standard)	Reference Standards Acyltransferase	Cardiovascular Disease Neurological Disease Metabolic Disease Cancer
GOAT-IN-1 (Standard) is the analytical standard of GOAT-IN-1 (HY-103479). This product is intended for research and analytical applications. GOAT-IN-1 is an inhibitor of ghrelin O-acyltransferase (GOAT), which could be useful for the prophylaxis or treatment of obesity, diabetes, hyperlipidemia, metabolic, non-alcoholic fatty liver, steatohepatitis, sarcopenia, appetite control, alcohol/narcotic dependence, Alzheimer’s disease, Parkinson’s disease, cerebrovascular dementia, cerebral apoplexy, cerebral infarction, cardic disease, some kind of tumors.

HY-B2185

Tipepidine citrate	Dopamine Receptor Potassium Channel AMPK	Neurological Disease Metabolic Disease Inflammation/Immunology
Tipepidine citrate is a non-narcotic antitussive agent. Tipepidine citrate reversibly inhibits dopamine D₂ receptor-mediated GIRK current (I_DA(GIRK)), thereby activating VTA dopamine neurons, with an IC₅₀ of 7.0 μM for I_DA(GIRK). Tipepidine activates AMPK. Tipepidine citrate has antidepressant-like effects. Tipepidine citrate enhances the analgesic effect of Carbamazepine (HY-B0246). Tipepidine citrate improves adipose tissue fibrosis and glucose intolerance in high-fat diet-induced obese mice .

HY-105628

Prodilidine CI-427	Others	Neurological Disease Inflammation/Immunology
Prodilidine (CI-427) is an orally active, pyrrolidine-derived non-narcotic pain inhibitor. Prodilidine exerts analgesic activity against various nociceptive stimuli, and shows no antipyretic, anti-inflammatory or respiratory depressive effects. Prodilidine fails to inhibit withdrawal symptoms of addictive agents in monkeys, but exhibits excitatory effects and enhances the crossed extensor reflex at toxic doses. Prodilidine is well absorbed from the gastrointestinal tract and metabolized via hepatic microsomal N-demethylation, displaying isomer-specific activity, toxicity and metabolic characteristics. Prodilidine can be used in research related to chronic pain (e.g., cancer-, musculoskeletal/arthritis-derived), traumatic pain and arthritic pain .

Cat. No.	Product Name	Category	Target	Chemical Structure

HY-B0264

Guaifenesin Guaiacol glyceryl ether; Guaiphenesin; Glycerol guaiacolate	Guaiacum officinale L. Natural Products other families Neurological Disease Classification of Application Fields Zygophyllaceae Plants Inflammation/Immunology Disease Research Fields Source Classification	Mucin
Guaifenesin (Guaiacol glyceryl ether), a constituent of guaiac resin from the wood of Guajacum officinale Linné, is an expectorant. Guaifenesin can alleviate cough discomfortby increasing sputum volume and decreasing its viscosity, thereby promoting effective cough .

HY-N7869

Celangulin VII	Structural Classification Terpenoids Celastraceae Celastrus angulatus Maxim. Plants Source Classification	Insecticide
Celangulin VII is a β-dihydroagarofuran sesquiterpene polyol ester present in the root bark of Celastrus angulatus. Celangulin VII exhibits insecticidal and narcotic activities against the 4th-instar larvae of Mythimna separata. Celangulin VII can be used in insecticide-related research .

Cat. No.	Product Name	Chemical Structure

HY-B0264S1

Guaifenesin-d5
Guaifenesin-d₅ is the deuterium labeled Guaifenesin. Guaifenesin (Guaiacol glyceryl ether), a constituent of guaiac resin from the wood of Guajacum officinale Linné, is an expectorant. Guaifenesin can alleviate cough discomfortby increasing sputum volume and decreasing its viscosity, thereby promoting effective cough. Guaifenesin also has narcotic effect .

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narcotic

Inhibitors & Agonists

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Isotope-Labeled Compounds

Natural
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