1. Cell Cycle/DNA Damage
    Epigenetics
  2. HDAC
  3. CXD101

CXD101 

Cat. No.: HY-100748 Purity: 99.14%
Handling Instructions

CXD101 is a class I-selective HDAC inhibitor (HDAC1 (IC50, 63 nM), HDAC2 (IC50, 570 nM), HDAC3 (IC50, 550 nM). CXD101 has no activity against HDAC class II.

For research use only. We do not sell to patients.

CXD101 Chemical Structure

CXD101 Chemical Structure

CAS No. : 934828-12-3

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 151 In-stock
Estimated Time of Arrival: December 31
1 mg USD 70 In-stock
Estimated Time of Arrival: December 31
5 mg USD 170 In-stock
Estimated Time of Arrival: December 31
10 mg USD 250 In-stock
Estimated Time of Arrival: December 31
50 mg USD 760 In-stock
Estimated Time of Arrival: December 31
100 mg USD 1070 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

Based on 1 publication(s) in Google Scholar

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Description

CXD101 is a class I-selective HDAC inhibitor (HDAC1 (IC50, 63 nM), HDAC2 (IC50, 570 nM), HDAC3 (IC50, 550 nM). CXD101 has no activity against HDAC class II[1].

IC50 & Target[1]

HDAC1

63 nM (IC50)

HDAC3

550 nM (IC50)

HDAC2

570 nM (IC50)

Clinical Trial
Molecular Weight

403.52

Formula

C₂₄H₂₉N₅O

CAS No.

934828-12-3

SMILES

O=C(NC1=C(N)C=CC=C1)C2=CC=C(C3CCN(CC4=CN(C)N=C4C)CC3)C=C2

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : ≥ 31 mg/mL (76.82 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.4782 mL 12.3910 mL 24.7819 mL
5 mM 0.4956 mL 2.4782 mL 4.9564 mL
10 mM 0.2478 mL 1.2391 mL 2.4782 mL
*Please refer to the solubility information to select the appropriate solvent.
References
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CXD101
Cat. No.:
HY-100748
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