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Art. -Nr.: HY-148137

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CB1 agonist 1

1 Cited Publications

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Based on 1 publication(s) in Google Scholar

CB1 agonist 1 (compound 22) is an agonist of CB1. CB1 agonist 1 shows affinity to CB1 receptor with an pIC₅₀ value of 5.7. CB1 agonist 1 can be used for the research of brain disorders.

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Reinheit: 99.84%
CAS. Nr.: 851212-80-1
Formel: C₂₄H₂₄N₂O₅S
Molecular Weight:452.52

Speicherung:

Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month

CB1 agonist 1 Chemical Structure

CAS. Nr.: 851212-80-1

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Biologische Aktivität
- Beschreibung
Chemical Information
Publications (1)
Lösungsmittel & Löslichkeit
- In Vitro
Reinheit & Dokumentation
Verweise
Help & FAQs
Classifications
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Biologische Aktivität

Beschreibung

CB1 agonist 1 (compound 22) is an agonist of CB1. CB1 agonist 1 shows affinity to CB1 receptor with an pIC₅₀ value of 5.7. CB1 agonist 1 can be used for the research of brain disorders^[1].

Alle Cannabinoid Receptor Isoform-spezifische Produkte anzeigen :

Chemical Information

CAS. Nr. 851212-80-1
Appearance Solid
Molecular Weight 452.52
Formel C₂₄H₂₄N₂O₅S
Color White to off-white
SMILES

O=C(C1=C(OC2=CC=CC=C2)C=CC=C1)NC3=CC=C(C)C(S(=O)(N4CCOCC4)=O)=C3
Versand

Room temperature in continental US; may vary elsewhere.

Speicherung

Powder	-20°C	3 years
In solvent	-80°C	6 months
	-20°C	1 month

Publications (1)

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Molecules

BI-5756 Reduces Graft-Versus-Host Disease Through CB1-Mediated Treg Upregulation. [Abstract]

2025 Aug 28;30(17):3517. PMID: 40942043

Lösungsmittel & Löslichkeit

In Vitro:

DMSO : 250 mg/mL (552.46 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

View the Complete Stock Solution Preparation Table

Preparing Stock Solutions

View the Complete Stock Solution Preparation Table

Concentration Solvent Mass

1 mg

5 mg

10 mg

Concentration

Solvent

Mass

1 mM

2.2098 mL

11.0492 mL

22.0985 mL

5 mM

0.4420 mL

2.2098 mL

4.4197 mL

10 mM

0.2210 mL

1.1049 mL

2.2098 mL

Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.

Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Molaritätsrechner

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Konzentration Konzentration

Volumen Volumen

Molecular Weight Molecular Weight

Verdünnungsrechner

Konzentration _{(Stammlösung)} × Volumen _{(Stammlösung)} = Konzentration _{(Ziellösung)} × Volumen _{(Ziellösung)}

Konzentration _{(Stammlösung)} Konzentration _{(Stammlösung)}

Volumen _{(Stammlösung)} Volumen _{(Stammlösung)}

Konzentration _{(Ziellösung)} Konzentration _{(Ziellösung)}

Volumen _{(Ziellösung)} Volumen _{(Ziellösung)}

Reinheit & Dokumentation

Select Batch:

Reinheit: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (269 KB)
SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

Verweise

[1]. Lambeng N, et al. Arylsulfonamides as a new class of cannabinoid CB1 receptor ligands: identification of a lead and initial SAR studies. Bioorg Med Chem Lett. 2007 Jan 1;17(1):272-7. [Content Brief]

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Complete Stock Solution Preparation Table

Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg
DMSO	1 mM	2.2098 mL	11.0492 mL	22.0985 mL	55.2462 mL
	5 mM	0.4420 mL	2.2098 mL	4.4197 mL	11.0492 mL
	10 mM	0.2210 mL	1.1049 mL	2.2098 mL	5.5246 mL
	15 mM	0.1473 mL	0.7366 mL	1.4732 mL	3.6831 mL
	20 mM	0.1105 mL	0.5525 mL	1.1049 mL	2.7623 mL
	25 mM	0.0884 mL	0.4420 mL	0.8839 mL	2.2098 mL
	30 mM	0.0737 mL	0.3683 mL	0.7366 mL	1.8415 mL
	40 mM	0.0552 mL	0.2762 mL	0.5525 mL	1.3812 mL
	50 mM	0.0442 mL	0.2210 mL	0.4420 mL	1.1049 mL
	60 mM	0.0368 mL	0.1842 mL	0.3683 mL	0.9208 mL
	80 mM	0.0276 mL	0.1381 mL	0.2762 mL	0.6906 mL
	100 mM	0.0221 mL	0.1105 mL	0.2210 mL	0.5525 mL

Keywords

CB1 agonist 1

1 Cited Publications

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Biologische Aktivität
- Beschreibung
Chemical Information
Publications (1)
Lösungsmittel & Löslichkeit
- In Vitro
Reinheit & Dokumentation
Verweise

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CB1 agonist 1

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Membrane Receptor-targeted Compound Library

Bioactive Compound Library Max

MCE Bioactive Compound Library

Bioactive Compound Library

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Publications Citing Use of MedChemExpress (MCE) CB1 agonist 1

Alle Cannabinoid Receptor Isoform-spezifische Produkte anzeigen

Biologische Aktivität

Chemical Information

Publications (1)

Lösungsmittel & Löslichkeit

Reinheit & Dokumentation

Verweise

Help & FAQs

Complete Stock Solution Preparation Table

CB1 agonist 1

GPCR/G Protein Compound Library

Neuronal Signaling Compound Library

Anti-Prostate Cancer Compound Library

Pain-Related Compound Library

Membrane Protein-targeted Compound Library

Membrane Receptor-targeted Compound Library

Bioactive Compound Library Max

MCE Bioactive Compound Library

Bioactive Compound Library

High-Throughput Bioactive Compound Library

Lactylation Compound Library

Publications Citing Use of MedChemExpress (MCE) CB1 agonist 1

Alle Cannabinoid Receptor Isoform-spezifische Produkte anzeigen

Biologische Aktivität

Chemical Information

Publications (1)

Lösungsmittel & Löslichkeit

Reinheit & Dokumentation

Verweise

Help & FAQs

Complete Stock Solution Preparation Table

CB1 agonist 1 Related Classifications

HY-148137 Related Classifications