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Referencia número: HY-162892

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BRD4-IN-9

BRD4-IN-9 is an orally active BRD4 inhibitor with an IC₅₀ value of 9.4 nM. BRD4-IN-9 can suppress tumor growth in a mouse melanoma xenograft model.

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No. CAS: 2468959-08-0
Fòrmula: C₂₄H₂₃N₃O₃
Peso molecular:401.46

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (267 KB)

BRD4-IN-9 Chemical Structure

No. CAS: 2468959-08-0

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Actividad biológica

Descripciòn

BRD4-IN-9 is an orally active BRD4 inhibitor with an IC₅₀ value of 9.4 nM. BRD4-IN-9 can suppress tumor growth in a mouse melanoma xenograft model^[1].

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Chemical Information

No. CAS 2468959-08-0
Peso molecular 401.46
Fòrmula C₂₄H₂₃N₃O₃
SMILES

CN(C(C=C1)=O)C=C1C2=CC=C(N=C(C3CCOCC3)N4)C4=C2OC5=CC=CC=C5
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureza y Documentación

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Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (267 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Horai Y, et al. A novel 7-phenoxy-benzimidazole derivative as a potent and orally available BRD4 inhibitor for the treatment of melanoma. Bioorg Med Chem. 2024 Oct 1;112:117882. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Actividad biológica
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BRD4-IN-9

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