Amperozide
Based on 1 Customer Validation
Amperozide is an atypical antipsychotic that acts as an antagonist of the 5-HT2 receptor with a Ki value of 26 nM. Amperozide has a low affinity for D2 receptors.
For research use only. We do not sell to patients.
- Purity: 99.10%
- CAS No.: 75558-90-6
- Formula: C23H29F2N3O
- Molecular Weight:401.49
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Storage:
4°C, protect from light
* In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
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Solvent & Solubility
- Purity & Documentation
- References
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Help & FAQs
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All 5-HT Receptor Isoforms
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Biological Activity
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5-HT2A Receptor 26 nM (Ki) |
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HepG2 | IC50 |
95 μM
Compound: Amperozide
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Cytotoxicity activity against human HepG2 cells after 24 hrs
Cytotoxicity activity against human HepG2 cells after 24 hrs
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[PMID: 20547797] |
Chemical Information
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CAS No. 75558-90-6
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Appearance Solid
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Molecular Weight 401.49
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Formula C23H29F2N3O
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Color White to off-white
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SMILES
O=C(NCC)N1CCN(CC1)CCCC(C2=CC=C(C=C2)F)C3=CC=C(C=C3)F
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
4°C, protect from light
* In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
Solvent & Solubility
DMSO : 125 mg/mL (311.34 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (267 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.4907 mL | 12.4536 mL | 24.9072 mL | 62.2681 mL |
| 5 mM | 0.4981 mL | 2.4907 mL | 4.9814 mL | 12.4536 mL | |
| 10 mM | 0.2491 mL | 1.2454 mL | 2.4907 mL | 6.2268 mL | |
| 15 mM | 0.1660 mL | 0.8302 mL | 1.6605 mL | 4.1512 mL | |
| 20 mM | 0.1245 mL | 0.6227 mL | 1.2454 mL | 3.1134 mL | |
| 25 mM | 0.0996 mL | 0.4981 mL | 0.9963 mL | 2.4907 mL | |
| 30 mM | 0.0830 mL | 0.4151 mL | 0.8302 mL | 2.0756 mL | |
| 40 mM | 0.0623 mL | 0.3113 mL | 0.6227 mL | 1.5567 mL | |
| 50 mM | 0.0498 mL | 0.2491 mL | 0.4981 mL | 1.2454 mL | |
| 60 mM | 0.0415 mL | 0.2076 mL | 0.4151 mL | 1.0378 mL | |
| 80 mM | 0.0311 mL | 0.1557 mL | 0.3113 mL | 0.7784 mL | |
| 100 mM | 0.0249 mL | 0.1245 mL | 0.2491 mL | 0.6227 mL |
Amperozide Related Classifications
HY-121301 Related Classifications
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