4 Results for "

2,5-Dimethoxy-4-iodoamphetamine

" in MedChemExpress (MCE) Product Catalog:
Products (4)

4 Results for "2,5-Dimethoxy-4-iodoamphetamine" in MCE Product Catalog:

Referencia número: HY-P3567
No. CAS: 159600-82-5
Target:  

Melanocortin Receptor

Áreas de investigación:  

Neurological Disease

(p-Iodo-Phe7)-ACTH (4-10) is a adrenocorticotrophic hormone (ACTH) derivative, which is produced and secreted by the anterior pituitary gland. (p-Iodo-Phe7)-ACTH (4-10) serves as a melanocortin (MC) receptor antagonist and inhibits α-melanocyte-stimulating hormone (α-MSH)-induced excessive grooming behavior in rats .
loading...
    loading...
Referencia número: HY-P2434
No. CAS: 846569-60-6
Target:  

Somatostatin Receptor

Áreas de investigación:  

Neurological Disease Metabolic Disease Cancer

AP102 is a dual SSTR2/SSTR5-specific somatostatin analog (SSA). AP102 is a disulfide-bridged octapeptide SSA containing synthetic iodinated amino acids. AP102 binds with subnanomolar affinity to SSTR2 and SSTR5 (IC50: 0.63 and 0.65 nM, respectively). AP102 does not bind to SSTR1 or SSTR3. AP102 can be used for acromegaly and neuroendocrine tumors research .
loading...
    loading...
Referencia número: HY-121775
No. CAS: 846032-02-8
Target:  

Dopamine Receptor

Áreas de investigación:  

Neurological Disease

F-00217830 is an agonist ofDopamine D2 receptor. PF-00217830 inhibits of spontaneous locomotor activity and 2,5-dimethoxy-4-iodoamphetamine-induced head twitches in rats .
loading...
    loading...
Referencia número: HY-134483
No. CAS: 851375-22-9
Target:  

5-HT Receptor

Áreas de investigación:  

Neurological Disease

5-HT7/5-HT2A receptor antagonist 1 is a high-affinity, orally active, brain-penetrant 5-HT7 and 5-HT2A receptor ligand having a pKi = 8.1 at both receptors. 5-HT7/5-HT2A receptor antagonist 1 behaves as an antagonist in an in vitro functional assay for 5-HT2A and as an inverse agonist in an in vitro functional assay for 5-HT7. 5-HT7/5-HT2A receptor antagonist 1 blockade of 5-Carboxamidotryptamine (5-CT) (HY-135555) induced hypothermia in rats, and blockade of 2,5-dimethoxy-4-iodoamphetamine (DOI) induced head-twitches in mice. 5-HT7/5-HT2A receptor antagonist 1 occupied 5-HT2A receptor binding sites in the frontal cortex of the rat brain. 5-HT7/5-HT2A receptor antagonist 1 can be used for the study of Neurological diseases .
loading...
    loading...