846569-60-6
Chemical Structure
AP102
- No. CAS: 846569-60-6
- Formula:C50H66I2N12O10S2
- Molecular Weight:1313.07
InChIKey: ISZMJWBQCGWNNM-DQIXCUPKSA-N
SMILES: O=C(N[C@H](C(N[C@H](C(N1)=O)C(C)C)=O)CCCCN)[C@H](NC([C@@H](NC([C@H](CSSC[C@H]1C(N[C@H](C(N)=O)[C@H](O)C)=O)NC([C@H](N)CC(C=C2)=CC(I)=C2N)=O)=O)CC(C=C3)=CC(I)=C3O)=O)CC4=CNC5=CC=CC=C45
Biological Activity: AP102 is a dual SSTR2/SSTR5-specific somatostatin analog (SSA). AP102 is a disulfide-bridged octapeptide SSA containing synthetic iodinated amino acids. AP102 binds with subnanomolar affinity to SSTR2 and SSTR5 (IC50: 0.63 and 0.65 nM, respectively). AP102 does not bind to SSTR1 or SSTR3. AP102 can be used for acromegaly and neuroendocrine tumors research[1].
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AP102 | AP102 is a dual SSTR2/SSTR5-specific somatostatin analog (SSA). AP102 is a disulfide-bridged octapeptide SSA containing synthetic iodinated amino acids. AP102 binds with subnanomolar affinity to SSTR2 and SSTR5 (IC50: 0.63 and 0.65 nM, respectively). AP102 does not bind to SSTR1 or SSTR3. AP102 can be used for acromegaly and neuroendocrine tumors research. | |||||||||||||||||||||
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