4 Results for "

EphA2 agonist

" in MedChemExpress (MCE) Product Catalog:
Products (4)

4 Results for "EphA2 agonist" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-P10579
CAS No.: 2225868-19-7
Target:  

Ephrin Receptor

Research Areas:  

Cancer

123B9, a tumor-homing agent, is a potent and selective EphA2 agonist with a Kd value of 4.0 μM. 123B9 selectively targets the EphA2 tyrosine kinase receptor ligand-binding domain. 123B9 does not appreciably inhibit the ligand binding domains of the most closely related EphA3 and EphA4 receptors .
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Cat. No.: HY-147637
CAS No.: 2611459-57-3
Purity:  99.32%
Target:  

Ephrin Receptor

Research Areas:  

Cancer

EphA2 agonist 1 (Compound 7bg) is a potent EphA2 receptor agonist. EphA2 agonist 1 shows great potency and selectivity toward EphA2 overexpressed glioblastoma cells and stimulates EphA2 phosphorylation .
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Cat. No.: HY-146141
CAS No.: 2169273-66-7
Target:  

Ephrin Receptor

Research Areas:  

Cancer

EphA2 agonist 2 (Lead compound) is a selective EphA2 agonist with antitumor activities. EphA2 agonist 2 can cross the BBB .
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Cat. No.: HY-P11015
Target:  

Ephrin Receptor

Research Areas:  

Cancer

(123B9)2-Motif is a selective EphA2 receptor agonist (Kd=4.9 μM) that does not bind to EphA4. (123B9)2-Motif works by inducing EphA2 receptor phosphorylation and oligomerization, thereby promoting receptor activation and internalization. (123B9)2-Motif is primarily used in targeted drug delivery studies for cancers that overexpress EphA2, such as breast cancer, to reduce circulating tumor cells and inhibit metastasis .
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