1. Protein Tyrosine Kinase/RTK
  2. Ephrin Receptor
  3. EphA2 agonist 2

EphA2 agonist 2 

Cat. No.: HY-146141
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EphA2 agonist 2 (Lead compound) is a selective EphA2 agonist with antitumor activities. EphA2 agonist 2 can cross the BBB.

For research use only. We do not sell to patients.

EphA2 agonist 2 Chemical Structure

EphA2 agonist 2 Chemical Structure

CAS No. : 2169273-66-7

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Description

EphA2 agonist 2 (Lead compound) is a selective EphA2 agonist with antitumor activities. EphA2 agonist 2 can cross the BBB[1].

In Vitro

EphA2 agonist 2 (Lead compound) shows antiproliferation activity with IC50 values of 2.1 ± 1.05 μM and 5.2 ± 2.56 μM against U251 EphA2 overexpressed and U251 wild type cells, respectively[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

772.94

Formula

C40H56N10O6

CAS No.
SMILES

O=C(N1CCN(C2=NC(N)=C3C=C(OC)C(OC)=CC3=N2)CC1)CCCCCCCCCCC(N4CCN(C5=NC(N)=C6C=C(OC)C(OC)=CC6=N5)CC4)=O

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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
EphA2 agonist 2
Cat. No.:
HY-146141
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