(123B9)2-Motif
(123B9)2-Motif is a selective EphA2 receptor agonist (Kd=4.9 μM) that does not bind to EphA4. (123B9)2-Motif works by inducing EphA2 receptor phosphorylation and oligomerization, thereby promoting receptor activation and internalization. (123B9)2-Motif is primarily used in targeted drug delivery studies for cancers that overexpress EphA2, such as breast cancer, to reduce circulating tumor cells and inhibit metastasis.
For research use only. We do not sell to patients.
- Formula: C142H197Cl2F2N31O47
- Molecular Weight:3199.17
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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EPHA2 |
Chemical Information
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Molecular Weight 3199.17
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Formula C142H197Cl2F2N31O47
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)