1. Protein Tyrosine Kinase/RTK
  2. Ephrin Receptor
  3. EphA2 agonist 1

EphA2 agonist 1 

Cat. No.: HY-147637
Handling Instructions

EphA2 agonist 1 (Compound 7bg) is a potent EphA2 receptor agonist. EphA2 agonist 1 shows great potency and selectivity toward EphA2 overexpressed glioblastoma cells and stimulates EphA2 phosphorylation.

For research use only. We do not sell to patients.

EphA2 agonist 1 Chemical Structure

EphA2 agonist 1 Chemical Structure

CAS No. : 2611459-57-3

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Description

EphA2 agonist 1 (Compound 7bg) is a potent EphA2 receptor agonist. EphA2 agonist 1 shows great potency and selectivity toward EphA2 overexpressed glioblastoma cells and stimulates EphA2 phosphorylation[1].

IC50 & Target

EphA2[1]

In Vitro

EphA2 agonist 1 (Compound 7bg) inhibits cell proliferation with IC50 values of 1.90 ± 0.55 μM and 7.91 ± 2.28 μM against U251 EphA2 overexpressed and U251 wild type cells, respectively[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

1019.07

Formula

C50H58N12O12

CAS No.
SMILES

COC1=C(C=C2C(N=C(N=C2N)N3CCN(CC3)C(C4=CC(NC(OCCOCCOCCOC(NC5=CC=CC(C(N6CCN(CC6)C7=NC8=CC(OC)=C(C=C8C(N)=N7)OC)=O)=C5)=O)=O)=CC=C4)=O)=C1)OC

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
EphA2 agonist 1
Cat. No.:
HY-147637
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